TRIFLUOROMETHYLATED HETEROCYCLES FROM BETA-TRIFLUOROACETYL-LACTAMS AND BETA-TRIFLUOROBENZOLACTAMS

被引：40

作者：

BOUILLON, JP ^{[1
]}

ATES, C ^{[1
]}

JANOUSEK, Z ^{[1
]}

VIEHE, HG ^{[1
]}

机构：

[1] LAB CHIM ORGAN,PL L PASTEUR 1,B-1348 LOUVAIN,BELGIUM

来源：

TETRAHEDRON LETTERS | 1993年 / 34卷 / 32期

关键词：

D O I：

10.1016/S0040-4039(00)60679-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Trifluoromethyl substituted heterocycles have been prepared by condensation of the new beta-trifluoroacetyl-lactams 1 and -benzolactams 2 with methylhydrazine and benzamidine as bis-nucleophiles without opening of the lactam structure.

引用

页码：5075 / 5078

页数：4

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