STRUCTURAL BASIS FOR CHEMICAL INHIBITION OF CDK2, A CELL-CYCLE CONTROLLING PROTEIN-KINASE

被引:0
|
作者
SUNGHOU, K [1 ]
机构
[1] UNIV CALIF BERKELEY,BERKELEY,CA 94720
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
引用
收藏
页码:257 / MEDI
相关论文
共 50 条
  • [1] STRUCTURAL BASIS FOR ACTIVATION OF CDK2, A CELL-CYCLE KINASE
    KIM, SH
    FASEB JOURNAL, 1994, 8 (07): : A1322 - A1322
  • [2] REGULATION OF THE CELL-CYCLE BY THE CDK2 PROTEIN-KINASE IN CULTURED HUMAN FIBROBLASTS
    PAGANO, M
    PEPPERKOK, R
    LUKAS, J
    BALDIN, V
    ANSORGE, W
    BARTEK, J
    DRAETTA, G
    JOURNAL OF CELL BIOLOGY, 1993, 121 (01): : 101 - 111
  • [3] Structural basis for specificity and potency of a flavonoid inhibitor of human CDK2, a cell cycle kinase
    deAzevedo, WF
    MuellerDieckmann, HJ
    SchulzeGahmen, U
    Worland, PJ
    Sausville, E
    Kim, SH
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1996, 93 (07) : 2735 - 2740
  • [4] Structure-based inhibitor design for CDK2, a cell cycle controlling protein kinase
    Kim, SH
    PURE AND APPLIED CHEMISTRY, 1998, 70 (03) : 555 - 565
  • [5] CDK2 ENCODES A 33-KDA CYCLIN-A-ASSOCIATED PROTEIN-KINASE AND IS EXPRESSED BEFORE CDC2 IN THE CELL-CYCLE
    ELLEDGE, SJ
    RICHMAN, R
    HALL, FL
    WILLIAMS, RT
    LODGSON, N
    HARPER, JW
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1992, 89 (07) : 2907 - 2911
  • [6] Rapid adaptation to CDK2 inhibition exposes intrinsic cell-cycle plasticity
    Arora, Mansi
    Moser, Justin
    Hoffman, Timothy E.
    Watts, Lotte P.
    Min, Mingwei
    Musteanu, Monica
    Rong, Yao
    Ryland III, C.
    Nangia, Varuna
    Schneider, Jordan
    Sanclemente, Manuel
    Lapek, John
    Nguyen, Lisa
    Niessen, Sherry
    Dann, Stephen
    VanArsdale, Todd
    Barbacid, Mariano
    Miller, Nichol
    Spencer, Sabrina L.
    CELL, 2023, 186 (12) : 2628 - +
  • [7] CDK2 ENCODES A CYCLIN-A ASSOCIATED PROTEIN-KINASE HOMOLOG OF CDC2 AND IS EXPRESSED EARLIER IN THE CELL-CYCLE THAN IS CDC2
    HARPER, JW
    RICHMAN, R
    HALL, FL
    WILLIAMS, RT
    LODGSON, N
    ELLEDGE, SJ
    FASEB JOURNAL, 1992, 6 (01): : A39 - A39
  • [8] CHROMOSOMAL MAPPING OF HUMAN CDK2, CDK4, AND CDK5 CELL-CYCLE KINASE GENES
    DEMETRICK, DJ
    ZHANG, H
    BEACH, DH
    CYTOGENETICS AND CELL GENETICS, 1994, 66 (01): : 72 - 74
  • [9] REGULATION OF THE VERTEBRATE CELL-CYCLE BY THE CDC2 PROTEIN-KINASE
    DRAETTA, G
    BRIZUELA, L
    MORAN, B
    BEACH, D
    COLD SPRING HARBOR SYMPOSIA ON QUANTITATIVE BIOLOGY, 1988, 53 : 195 - 201
  • [10] Selective chemical inhibition as a tool to study Cdk1 and Cdk2 functions in the cell cycle
    Krasinska, Liliana
    Cot, Emilie
    Fisher, Daniel
    CELL CYCLE, 2008, 7 (12) : 1702 - 1708