A FACILE ONE-POT SYNTHESIS OF 5-TRIFLUOROMETHYLOXAZOLES AND 5-PERFLUOROALKYLOXAZOLES FROM N-ALKYL-N-ACYLAMINO ACIDS

被引：9
|
作者：
KAWASE, M
机构：
[1] Faculty of Pharmaceutical Sciences, Josai University, Sakado-shi, Saitama, 350-02
来源：
HETEROCYCLES | 1993年 / 36卷 / 11期
关键词：
D O I：
10.3987/COM-93-6508
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The reaction of N-acyl-N-benzyl-alpha-amino acids with trifluoroacetic or perfluorocarboxylic anhydride in the presence of pyridine affords 5-trifluoromethyl- or 5-perfluoroalkyloxazoles in high yields.
引用
收藏
页码：2441 / 2444
页数：4
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