THE SOLID-PHASE SYNTHESIS OF DIHYDROISOQUINOLINES AND TETRAHYDROISOQUINOLINES

被引：46

作者：

MEUTERMANS, WDF

ALEWOOD, PF

机构：

[1] Centre for Drug Design and Development, University of Queensland, Brisbane

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 42期

关键词：

D O I：

10.1016/0040-4039(95)01569-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Tetrahydroisoquinolines have been synthesised on Merrifield resin in good fields and high purity via the Bischler-Napieralski approach. A one pot multiple synthesis was developed and the reaction sequence monitored using ionspray mass spectrometry.

引用

页码：7709 / 7712

页数：4

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