THROMBOXANE RECEPTOR ANTAGONISM COMBINED WITH THROMBOXANE SYNTHASE INHIBITION .8. N-ALKYLATION OF INDOLE RING USING MITSUNOBU REACTION

被引：21

作者：

BHAGWAT, SS

GUDE, C

机构：

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 12期

关键词：

D O I：

10.1016/S0040-4039(00)73177-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Indole rings substituted with two electron withdrawing groups were alkylated on the nitrogen under Mitsunobu reaction conditions.

引用

页码：1847 / 1850

页数：4

共 4 条

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[3]

DANISHEFSKY S, 1981, TETRAHEDRON LETT, P3919

[4] STUDIES ON GELSEMIUM ALKALOIDS - TOTAL SYNTHESIS OF (+)-KOUMINE, (+)-TABERPSYCHINE, AND (+)-KOUMIDINE [J].

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