L-663,536 (MK-886) (3-[1-(4-CHLOROBENZYL)-3-T-BUTYL-THIO-5-ISOPROPYLINDOL-2-YL]-2,2-DIMETHYLPROPANOIC ACID), A NOVEL, ORALLY ACTIVE LEUKOTRIENE BIOSYNTHESIS INHIBITOR

被引：354

作者：

GILLARD, J

FORDHUTCHINSON, AW

CHAN, C

CHARLESON, S

DENIS, D

FOSTER, A

FORTIN, R

LEGER, S

MCFARLANE, CS

MORTON, H

PIECHUTA, H

RIENDEAU, D

ROUZER, CA

ROKACH, J

YOUNG, R

MACINTYRE, DE

PETERSON, L

BACH, T

EIERMANN, G

HOPPLE, S

HUMES, J

HUPE, L

LUELL, S

METZGER, J

MEURER, R

MILLER, DK

OPAS, E

PACHOLOK, S

机构：

[1] MERCK FROSST CTR THERAPEUT RES,DEPT PHARMACOL,POB 1005,POINTE CLAIRE H9R 4P8,QUEBEC,CANADA

[2] MERCK SHARP & DOHME RES LABS,DEPT BIOCHEM & INFLAMMAT,RAHWAY,NJ 07065

[3] MERCK FROSST CTR THERAPEUT RES,DEPT MED CHEM,POINT CLAIRE H9R 4P8,QUEBEC,CANADA

来源：

CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY | 1989年 / 67卷 / 05期

关键词：

D O I：

10.1139/y89-073

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：456 / 464

页数：9

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