SUPERACTIVE ANTINOCICEPTIVE PENTAPEPTIDE, (D-MET2,PRO5), ENKEPHALINAMIDE

被引：143

作者：

BAJUSZ, S ^{[1
]}

RONAI, AZ ^{[1
]}

SZEKELY, JI ^{[1
]}

GRAF, L ^{[1
]}

DUNAIKOVACS, Z ^{[1
]}

BERZETEI, I ^{[1
]}

机构：

[1] RES INST PHARMACEUT CHEM,H-1325 BUDAPEST,HUNGARY

来源：

FEBS LETTERS | 1977年 / 76卷 / 01期

关键词：

D O I：

10.1016/0014-5793(77)80127-0

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：91 / 92

页数：2

共 11 条

[1]

BAJUSZ S, 1976, ACTA BIOCHIM BIOPHYS, V11, P305

[2]

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[3] SYNTHESIS AND OPIOID ACTIVITIES OF STEREOISOMERS AND OTHER D-AMINO-ACID ANALOGS OF METHIONINE-ENKEPHALIN [J].

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KASTIN, AJ ;

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FERTEL, R ;

BERNTSON, GG ;

SANDMAN, CA .

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[4]

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[5] COMPARATIVE-STUDY ON ANALGESIC EFFECT OF MET5-ENKEPHALIN AND RELATED LIPOTROPIN FRAGMENTS [J].

GRAF, L ;

SZEKELY, JI ;

RONAI, AZ ;

DUNAIKOVACS, Z ;

BAJUSZ, S .

NATURE, 1976, 263 (5574) :240-241

[6] MODE OF DEACTIVATION OF ENKEPHALINS BY RAT AND HUMAN-PLASMA AND RAT-BRAIN HOMOGENATES [J].

HAMBROOK, JM ;

MORGAN, BA ;

RANCE, MJ ;

SMITH, CFC .

NATURE, 1976, 262 (5571) :782-783

[7] IDENTIFICATION OF 2 RELATED PENTAPEPTIDES FROM BRAIN WITH POTENT OPIATE AGONIST ACTIVITY [J].

HUGHES, J ;

SMITH, TW ;

KOSTERLITZ, HW ;

FOTHERGILL, LA ;

MORGAN, BA ;

MORRIS, HR .

NATURE, 1975, 258 (5536) :577-579

[8] D-ALA2-MET-ENKEPHALINAMIDE - POTENT, LONG-LASTING SYNTHETIC PENTAPEPTIDE ANALGESIC [J].

PERT, CB ;

PERT, A ;

CHANG, JK ;

FONG, BTW .

SCIENCE, 1976, 194 (4262) :330-332

[9]

SZEKELY JI, 1977, EXPERIENTIA, V33, P54

[10]

TSENG LF, 1976, NATURE, V263, P239, DOI 10.1038/263239a0

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