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- [31] The first total synthesis of (±)-arisugacin A, a potent, orally bioavailable inhibitor of acetylcholinesteraseORGANIC LETTERS, 2002, 4 (03) : 367 - 369Sunazuka, T论文数: 0 引用数: 0 h-index: 0机构: Kitasato Univ, Kitasato Inst, Minato Ku, Tokyo 1088642, JapanHanda, M论文数: 0 引用数: 0 h-index: 0机构: Kitasato Univ, Kitasato Inst, Minato Ku, Tokyo 1088642, JapanNagai, K论文数: 0 引用数: 0 h-index: 0机构: Kitasato Univ, Kitasato Inst, Minato Ku, Tokyo 1088642, JapanShirahata, T论文数: 0 引用数: 0 h-index: 0机构: Kitasato Univ, Kitasato Inst, Minato Ku, Tokyo 1088642, JapanHarigaya, Y论文数: 0 引用数: 0 h-index: 0机构: Kitasato Univ, Kitasato Inst, Minato Ku, Tokyo 1088642, JapanOtoguro, K论文数: 0 引用数: 0 h-index: 0机构: Kitasato Univ, Kitasato Inst, Minato Ku, Tokyo 1088642, JapanKuwajima, I论文数: 0 引用数: 0 h-index: 0机构: Kitasato Univ, Kitasato Inst, Minato Ku, Tokyo 1088642, JapanOmura, S论文数: 0 引用数: 0 h-index: 0机构: Kitasato Univ, Kitasato Inst, Minato Ku, Tokyo 1088642, Japan
- [32] Discovery of potent, orally bioavailable protease-activated receptor 4 antagonistsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250Marinier, Anne论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaBanville, Jacques论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaBird, Eileen论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaCallejo, Mario论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaDeon, Daniel论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaDube, Laurence论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaGagnon, Marc论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaGiancarli, Mary论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaGuy, Julia论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaHarper, Tim论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaLam, Patrick论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaLavallee, Jean-Francois论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaLawrence, Michael论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaMartel, Alain论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaMiller, Michael论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaO'Grady, Harold论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaPosy, Shoshana论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaPriestley, Scott论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaRemillard, Roger论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaRuediger, Edward论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaTremblay, Francois论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaWatson, Carol论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaWong, Pancras论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaYang, Jing论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaBouvier, Michel论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaSeiffert, Dietmar论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, CanadaWexler, Ruth论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Cardiovasc Res, Hopewell, NJ USA Univ Montreal, Inst Res Immunol & Canc, Montreal, PQ, Canada
- [33] Identification of an Orally Bioavailable, Potent, and Selective Inhibitor of GlyT1ACS MEDICINAL CHEMISTRY LETTERS, 2010, 1 (07): : 350 - 354Blackaby, Wesley P.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandLewis, Richard T.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandThomson, Joanne L.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandJennings, Andrew S. R.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandGoodacre, Simon C.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandStreet, Leslie J.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandMacLeod, Angus M.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandPike, Andrew论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandWood, Suzanne论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandThomas, Steve论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandBrown, Terry A.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandSmith, Alison论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandPillai, Gopalan论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandAlmond, Sarah论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandGuscott, Martin R.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandBurns, H. Donald论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandEng, Waisi论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandRyan, Christine论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandCook, Jacquelynn论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, EnglandHamill, Terence G.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA 19486 USA Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Harlow CM20 2QR, Essex, England
- [34] Discovery of PF-04449913, a Potent and Orally Bioavailable Inhibitor of SmoothenedACS MEDICINAL CHEMISTRY LETTERS, 2012, 3 (02): : 106 - 111Munchhof, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Michael J Munchhof LLC, Salem, CT 06420 USA Michael J Munchhof LLC, Salem, CT 06420 USALi, Qifang论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton, CT 06340 USA Michael J Munchhof LLC, Salem, CT 06420 USAShavnya, Andrei论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton, CT 06340 USA Michael J Munchhof LLC, Salem, CT 06420 USABorzillo, Gary V.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton, CT 06340 USA Michael J Munchhof LLC, Salem, CT 06420 USABoyden, Tracey L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton, CT 06340 USA Michael J Munchhof LLC, Salem, CT 06420 USAJones, Christopher S.论文数: 0 引用数: 0 h-index: 0机构: Michael J Munchhof LLC, Salem, CT 06420 USALaGreca, Susan D.论文数: 0 引用数: 0 h-index: 0机构: INC Res, Old Lyme, CT 06371 USA Michael J Munchhof LLC, Salem, CT 06420 USAMartinez-Alsina, Luis论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton, CT 06340 USA Michael J Munchhof LLC, Salem, CT 06420 USAPatel, Nandini论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton, CT 06340 USA Michael J Munchhof LLC, Salem, CT 06420 USAPelletier, Kathleen论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton, CT 06340 USA Michael J Munchhof LLC, Salem, CT 06420 USAReiter, Larry A.论文数: 0 引用数: 0 h-index: 0机构: Reiter MedChem, Mystic, CT 06355 USA Michael J Munchhof LLC, Salem, CT 06420 USARobbins, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Princeton, NJ 08540 USA Michael J Munchhof LLC, Salem, CT 06420 USATkalcevic, George T.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Groton, CT 06340 USA Michael J Munchhof LLC, Salem, CT 06420 USA
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