SYNTHESIS AND STUDY OF A NON-MACROCYCLIC FK506 DERIVATIVE

被引:9
作者
TEAGUE, SJ
COOPER, ME
DONALD, DK
FURBER, M
机构
[1] Fisons plc, Pharmaceuticals Division, Loughborough, LE11 0RH, Bakewell Road
关键词
D O I
10.1016/S0960-894X(01)80570-9
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
The affinity of a non macrocyclic analogue of FK506 for the immunophilin FKBP12 was The affinity of this analogue/FKBP12 complex for calcineurin was studied.
引用
收藏
页码:1581 / 1584
页数:4
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