MUSCARINIC M2 RECEPTORS IN BOVINE TRACHEAL SMOOTH-MUSCLE - DISCREPANCIES BETWEEN BINDING AND FUNCTION

被引:159
|
作者
ROFFEL, AF [1 ]
ELZINGA, CRS [1 ]
VANAMSTERDAM, RGM [1 ]
DEZEEUW, RA [1 ]
ZAAGSMA, J [1 ]
机构
[1] UNIV GRONINGEN,DEPT ANALYT CHEM & TOXICOL,9713 AW GRONINGEN,NETHERLANDS
关键词
D O I
10.1016/0014-2999(88)90589-4
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:73 / 82
页数:10
相关论文
共 50 条
  • [1] SUBTYPES OF MUSCARINIC RECEPTORS IN BOVINE TRACHEAL SMOOTH-MUSCLE
    ROBERTS, MF
    ROETS, EA
    BURVENICH, C
    FASEB JOURNAL, 1992, 6 (04): : A1294 - A1294
  • [2] Effects of fenoterol on β-adrenoceptor and muscarinic M2 receptor function in bovine tracheal smooth muscle
    De Vries, B
    Roffel, AF
    Kooistra, JM
    Meurs, H
    Zaagsma, J
    EUROPEAN JOURNAL OF PHARMACOLOGY, 2001, 419 (2-3) : 253 - 259
  • [3] M2 muscarinic receptors inhibit forskolin -: but not isoproterenol-mediated relaxation in bovine tracheal smooth muscle
    Ostrom, RS
    Ehlert, FJ
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1998, 286 (01): : 234 - 242
  • [4] ALLOSTERIC INTERACTIONS OF 3 MUSCARINE ANTAGONISTS AT BOVINE TRACHEAL SMOOTH-MUSCLE AND CARDIAC M2 RECEPTORS
    ROFFEL, AF
    ELZINGA, CRS
    MEURS, H
    ZAAGSMA, J
    EUROPEAN JOURNAL OF PHARMACOLOGY-MOLECULAR PHARMACOLOGY SECTION, 1989, 172 (01): : 61 - 70
  • [5] Studies on muscarinic M2 receptors in smooth muscle
    Mitchelson, F
    Shen, A
    PROCEEDINGS OF THE FORTY-SECOND ANNUAL MEETING OF THE WESTERN PHARMACOLOGY SOCIETY, 1999, 42 : 109 - 110
  • [6] AFDX-116 DISCRIMINATES BETWEEN MUSCARINIC M2 RECEPTORS OF THE HEART AND THE IRIS SMOOTH-MUSCLE
    HONKANEN, RE
    ABDELLATIF, AA
    MOLECULAR AND CELLULAR BIOCHEMISTRY, 1988, 82 (1-2) : 131 - 135
  • [7] EXPRESSION OF MUSCARINIC M2 RECEPTORS IN CULTURED HUMAN AIRWAY SMOOTH-MUSCLE CELLS
    WIDDOP, S
    DAYKIN, K
    HALL, IP
    AMERICAN JOURNAL OF RESPIRATORY CELL AND MOLECULAR BIOLOGY, 1993, 9 (05) : 541 - 546
  • [8] Stimulation of muscarinic M2 receptors inhibits atrial natriuretic peptide-mediated relaxation in bovine tracheal smooth muscle
    Tsutomu Nakahara
    Motonari Yunoki
    Akiko Mitani
    Kenji Sakamoto
    Kunio Ishii
    Naunyn-Schmiedeberg's Archives of Pharmacology, 2002, 366 : 376 - 379
  • [9] Stimulation of muscarinic M2 receptors inhibits atrial natriuretic peptide-mediated relaxation in bovine tracheal smooth muscle
    Nakahara, T
    Yunoki, M
    Mitani, A
    Sakamoto, K
    Ishii, K
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 2002, 366 (04) : 376 - 379
  • [10] M2 AND M3-MUSCARINIC-RECEPTORS COEXIST IN CANINE COLONIC CIRCULAR SMOOTH-MUSCLE
    ZHANG, L
    BUXTON, ILO
    FASEB JOURNAL, 1991, 5 (06): : A1586 - A1586