INHIBITION OF CYP1A, CYP2B, AND CYP3A ACTIVITIES BY 5HT3 ANTAGONISTS

被引:0
作者
GAN, LS [1 ]
BOEHLERT, C [1 ]
THAKKER, D [1 ]
SERABJITSINGH, C [1 ]
机构
[1] GLAXO RES INST,DEPT DRUG METAB,RES TRIANGLE PK,NC 27709
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:A1248 / A1248
页数:1
相关论文
共 50 条
[31]   OMEPRAZOLE AND LANSOPRAZOLE ARE MIXED INDUCERS OF CYP1A AND CYP3A IN HUMAN HEPATOCYTES IN PRIMARY CULTURE [J].
CURIPEDROSA, R ;
DAUJAT, M ;
PICHARD, L ;
OURLIN, JC ;
CLAIR, P ;
GERVOT, L ;
LESCA, P ;
DOMERGUE, J ;
JOYEUX, H ;
FOURTANIER, G ;
MAUREL, P .
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1994, 269 (01) :384-392
[32]   CYP1A and CYP3A induction in cryopreserved Cynomolgus monkey hepatocytes pooled from multiple donors [J].
Doshi, Utkarsh ;
Yang, Qian ;
Li, Nicole ;
Li, Albert ;
Seagrave, JeanClare .
DRUG METABOLISM REVIEWS, 2011, 43 :101-101
[33]   Effects of alkylphenols on CYP1A and CYP3A expression in first spawning Atlantic cod (Gadus morhua) [J].
Hasselberg, L ;
Meier, S ;
Svardal, A ;
Hegelund, T ;
Celander, MC .
AQUATIC TOXICOLOGY, 2004, 67 (04) :303-313
[34]   INDUCTION OF THE HEPATIC CYP2B AND CYP3A ENZYMES BY THE PROESTROGENIC PESTICIDE METHOXYCHLOR AND BY DDT IN THE RAT - EFFECTS ON METHOXYCHLOR METABOLISM [J].
LI, HC ;
DEHAL, SS ;
KUPFER, D .
JOURNAL OF BIOCHEMICAL TOXICOLOGY, 1995, 10 (01) :51-61
[35]   Effect of fluvoxamine therapy on the activities of CYP1A2, CYP2D6, and CYP3A as determined by phenotyping [J].
Kashuba, ADM ;
Nafziger, AN ;
Kearns, GL ;
Leeder, JS ;
Gotschall, R ;
Rocci, ML ;
Kulawy, RW ;
Beck, DJ ;
Bertino, JS .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1998, 64 (03) :257-268
[36]   Exploring QSARs for binding affinity of azoles with CYP2B and CYP3A enzymes using GFA and G/PLS techniques [J].
Roy, Kunal ;
Roy, Partha Pratim .
CHEMICAL BIOLOGY & DRUG DESIGN, 2008, 71 (05) :464-473
[37]   CYP3A probes can quantitatively predict the in vivo kinetics of other CYP3A substrates and can accurately assess CYP3A induction and inhibition [J].
Kharasch, ED ;
Thummel, KE ;
Watkins, PB .
MOLECULAR INTERVENTIONS, 2005, 5 (03) :151-+
[38]   Sex and CYP3A5 genotype influence total CYP3A activity: high CYP3A activity and a unique distribution of CYP3A5 variant alleles in Ethiopians [J].
E Gebeyehu ;
E Engidawork ;
A Bijnsdorp ;
A Aminy ;
U Diczfalusy ;
E Aklillu .
The Pharmacogenomics Journal, 2011, 11 :130-137
[39]   Sex and CYP3A5 genotype influence total CYP3A activity: high CYP3A activity and a unique distribution of CYP3A5 variant alleles in Ethiopians [J].
Gebeyehu, E. ;
Engidawork, E. ;
Bijnsdorp, A. ;
Aminy, A. ;
Diczfalusy, U. ;
Aklillu, E. .
PHARMACOGENOMICS JOURNAL, 2011, 11 (02) :130-137
[40]   Effects of administration of the chemoprotective agent oltipraz on CYP1A and CYP2B in rat liver and rat hepatocytes in culture [J].
Langouet, S ;
Maheo, K ;
Berthou, F ;
Morel, F ;
LagadicGossman, D ;
Glaise, D ;
Coles, B ;
Ketterer, B ;
Guillouzo, A .
CARCINOGENESIS, 1997, 18 (07) :1343-1349