ENHANCEMENT OF SOLUBILITY, DISSOLUTION RATE, AND ORAL BIOAVAILABILITY OF RS-82856 BY COMPLEX-FORMATION WITH CYCLODEXTRINS

被引：4
|
作者：
YU, CD
SWEETANA, SA
CHU, NI
LEE, GJL
MASSEY, IJ
机构：
[1] SYNTEX RES CORP,INST PHARMACOL & DRUG METAB,PALO ALTO,CA 94304
[2] SYNTEX RES CORP,INST PHARMACEUT SCI,PALO ALTO,CA 94304
来源：
DRUG DEVELOPMENT AND INDUSTRIAL PHARMACY | 1989年 / 15卷 / 04期
关键词：
D O I：
10.3109/03639048909040233
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：609 / 620
页数：12
相关论文
共 34 条
  • [1] Studies on Enhancement of Solubility Dissolution Rate and Bioavailability of Glipizide by Complexation with β-Cyclodextrin
    Chowdary, K. P. R.
    Raga, Sunil
    ASIAN JOURNAL OF CHEMISTRY, 2012, 24 (04) : 1693 - 1697
  • [2] Solubility, Dissolution Rate and Bioavailability Enhancement of Irbesartan by Solid Dispersion Technique
    Boghra, Rikisha Jaysukhbhai
    Kothawade, Pranita Chandrakant
    Belgamwar, Veena Shailendra
    Nerkar, Pankaj Padmakar
    Tekade, Avinash Ramrao
    Surana, Sanjay Javerilal
    CHEMICAL & PHARMACEUTICAL BULLETIN, 2011, 59 (04) : 438 - 441
  • [3] Potential of erlotinib cyclodextrin nanosponge complex to enhance solubility, dissolution rate, in vitro cytotoxicity and oral bioavailability
    Dora, Chander Parkash
    Trotta, Francesco
    Kushwah, Varun
    Devasari, Naresh
    Singh, Charan
    Suresh, Sarasija
    Jain, Sanyog
    CARBOHYDRATE POLYMERS, 2016, 137 : 339 - 349
  • [4] Enhancement of The Solubility and The Dissolution Rate of Oral Nimodipine Formulation with Solid Dispersion
    Ellakwa, Takwa E.
    Ellakwa, Doha E.
    EGYPTIAN JOURNAL OF CHEMISTRY, 2021, 64 (02): : 721 - 728
  • [5] SOLUBILITY ENHANCEMENT OF NUCLEOSIDES AND STRUCTURALLY RELATED-COMPOUNDS BY COMPLEX-FORMATION
    CHEN, AX
    ZITO, SW
    NASH, RA
    PHARMACEUTICAL RESEARCH, 1994, 11 (03) : 398 - 401
  • [6] Bioavailability Enhancement of Artemether and Lumefantrine by Improving Solubility and Dissolution Rate using Solid Dispersion Technique
    Charde, Yogita M.
    Avari, Jasmine G.
    INDIAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2021, 83 (04) : 808 - 822
  • [7] Enhancement of solubility, dissolution rate and bioavailability of atorvastatin using solid lipid: in vitro and in vivo characterization
    Pandit A.P.
    Chavan T.T.
    Khandelwal K.R.
    Journal of Pharmaceutical Investigation, 2015, 45 (6) : 503 - 513
  • [8] Electrosprayed Polymeric Nanospheres for Enhanced Solubility, Dissolution Rate, Oral Bioavailability and Antihyperlipidemic Activity of Bezafibrate
    Sun, Ru
    Shen, Chengwu
    Shafique, Shumaila
    Mustapha, Omer
    Hussain, Talib
    Khan, Ikram Ullah
    Mehmood, Yasir
    Anwer, Khaleeq
    Shahzad, Yasser
    Yousaf, Abid Mehmood
    INTERNATIONAL JOURNAL OF NANOMEDICINE, 2020, 15 : 705 - 715
  • [9] Fabrication of fenofibrate nanocrystals by probe sonication method for enhancement of dissolution rate and oral bioavailability
    Ige, Pradum Pundlikrao
    Baria, Rohan K.
    Gattani, Surendra G.
    COLLOIDS AND SURFACES B-BIOINTERFACES, 2013, 108 : 366 - 373
  • [10] Biodegradable Porous Starch Spheres as a Novel Carrier for Enhancement of Dissolution Rate and Oral Bioavailability of Itraconazole
    Pawar, Jaywant
    Ali, Meer Tarique
    Fule, Ritesh
    Moravkar, Kailas
    Seervi, Madhaysingh
    Sathaye, Sadhana
    Amin, Purnima
    CURRENT DRUG DELIVERY, 2017, 14 (07) : 944 - 954
1234