PARTITION-COEFFICIENT AS A GUIDE TO THE DEVELOPMENT OF RADIOSENSITIZERS WHICH ARE LESS TOXIC THAN MISONIDAZOLE

被引:202
作者
BROWN, JM [1 ]
WORKMAN, P [1 ]
机构
[1] MED SCH CAMBRIDGE,MRC,CLIN ONCOL & RADIOTHERAPEUT UNIT,CAMBRIDGE,ENGLAND
关键词
D O I
10.2307/3575246
中图分类号
Q [生物科学];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:171 / 190
页数:20
相关论文
共 31 条
[11]  
CURRY SH, 1977, DRUG DISPOSITION PHA
[12]   RADIOSENSITIZATION OF SOLID TUMORS BY NITROIMIDAZOLES [J].
DENEKAMP, J ;
FOWLER, JF .
INTERNATIONAL JOURNAL OF RADIATION ONCOLOGY BIOLOGY PHYSICS, 1978, 4 (1-2) :143-151
[13]   CLINICAL TESTING OF RADIOSENSITIZER RO 07-0582 - EXPERIENCE WITH MULTIPLE DOSES [J].
DISCHE, S ;
SAUNDERS, MI ;
LEE, ME ;
ADAMS, GE ;
FLOCKHART, IR .
BRITISH JOURNAL OF CANCER, 1977, 35 (05) :567-579
[14]  
GRIFFIN JW, 1979, NEUROTOXICOLOGY, V1, P299
[15]   RADIOSENSITIZATION BY MISONIDAZOLE (RO 07-0582) - IMPORTANCE OF TIMING AND TUMOR CONCENTRATION OF SENSITIZER [J].
MCNALLY, NJ ;
DENEKAMP, J ;
SHELDON, P ;
FLOCKHART, IR ;
STEWART, FA .
RADIATION RESEARCH, 1978, 73 (03) :568-580
[16]  
MELLET LB, 1974, ANTINEOPLASTIC IMM 1, P330
[17]  
RAUTH AM, 1978, BRIT J CANCER, V37, P202
[18]  
ROCKWELL SC, 1972, J NATL CANCER I, V49, P735
[19]  
SOLOWAY AH, 1960, J PHARMACOL EXP THER, V129, P310
[20]   CORRELATION OF DRUG PENETRATION OF BRAIN AND CHEMICAL STRUCTURE [J].
SOLOWAY, AH .
SCIENCE, 1958, 128 (3338) :1572-1574