SOLID-PHASE SYNTHESIS OF PHOSPHONOPEPTIDES

被引：21

作者：

CAMPAGNE, JM ^{[1
]}

COSTE, J ^{[1
]}

JOUIN, P ^{[1
]}

机构：

[1] CNRS,INSERM,CTR PHARMACOL ENDOCRINOL,F-34094 MONTPELLIER 5,FRANCE

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 12期

关键词：

D O I：

10.1016/0040-4039(95)00224-Z

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A solid phase synthesis of a phosphonopeptide is described, in which a type 1 aminophosphonate with a free phosphonic acid was coupled just like an amino acid, using BOP as reagent.

引用

页码：2079 / 2082

页数：4

共 12 条

[1] EVALUATION OF INTRINSIC BINDING-ENERGY FROM A HYDROGEN-BONDING GROUP IN AN ENZYME-INHIBITOR [J].

BARTLETT, PA ;

MARLOWE, CK .

SCIENCE, 1987, 235 (4788) :569-571

[2] POTENT INHIBITION OF PEPSIN AND PENICILLOPEPSIN BY PHOSPHORUS-CONTAINING PEPTIDE ANALOGS [J].

BARTLETT, PA ;

HANSON, JE ;

GIANNOUSIS, PP .

JOURNAL OF ORGANIC CHEMISTRY, 1990, 55 (26) :6268-6274

[3] 1-AMINOALKYLPHOSPHONOUS ACIDS .1. ISOSTERES OF THE PROTEIN AMINO-ACIDS [J].

BAYLIS, EK ;

CAMPBELL, CD ;

DINGWALL, JG .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1984, (12) :2845-2853

[4] SYNTHESIS OF MIXED PHOSPHONATE DIESTER ANALOGS OF DIPEPTIDES USING BOP OR PYBOP REAGENTS [J].

CAMPAGNE, JM ;

COSTE, J ;

JOUIN, P .

TETRAHEDRON LETTERS, 1993, 34 (42) :6743-6744

[5] SOLID-PHASE SYNTHESIS OF PHOSPHINIC PEPTIDES [J].

CAMPAGNE, JM ;

COSTE, J ;

GUILLOU, L ;

HEITZ, A ;

JOUIN, P .

TETRAHEDRON LETTERS, 1993, 34 (26) :4181-4184

[6] SOLID-PHASE SYNTHESIS OF PEPTIDYLPHOSPHONATES [J].

CAMPBELL, DA ;

BERMAK, JC .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1994, 116 (13) :6039-6040

[7]

Guo Jincan, 1994, Journal of the American Chemical Society, V116, P6062, DOI 10.1021/ja00093a002

[8] CHARACTERIZATION OF A MONOCLONAL-ANTIBODY PRODUCED IN AN ATTEMPT TO MIMIC THE ACTIVE-SITE OF HIV ASPARTYL PROTEASE USING HAPTENS BASED ON INHIBITOR MODELS [J].

HANIN, V ;

CAMPAGNE, JM ;

DOMINICE, C ;

MANI, JC ;

DUFOUR, MN ;

JOUIN, P ;

PAU, B .

JOURNAL OF IMMUNOLOGICAL METHODS, 1994, 173 (02) :139-147

[9]

MERY J, 1992, PEPTIDE RES, V5, P233

[10]

MERY J, 1993, INT J PEPT PROT RES, V42, P44

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