POSITION-5 AT THE OXOTREMORINE SKELETON AS THE STEERING POSITION FOR ACTIVITY AT THE MUSCARINIC RECEPTORS

被引：10
作者：
AMSTUTZ, R
CLOSSE, A
GMELIN, G
机构：
来源：
HELVETICA CHIMICA ACTA | 1987年 / 70卷 / 08期
关键词：
D O I：
10.1002/hlca.19870700827
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
引用
收藏
页码：2232 / 2244
页数：13
相关论文
共 22 条
[1]   STEREOSELECTIVITY OF MUSCARINIC RECEPTORS INVIVO AND INVITRO FOR OXOTREMORINE ANALOGS - N-[4-(TERTIARY AMINO)-2-BUTYNYL]-5-METHYL-2-PYRROLIDONES [J].
AMSTUTZ, R ;
RINGDAHL, B ;
KARLEN, B ;
ROCH, M ;
JENDEN, DJ .
JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (12) :1760-1765
[2]   THE EFFECT OF MCN-A-343 ON MUSCARINIC RECEPTORS IN THE CEREBRAL-CORTEX AND HEART [J].
BIRDSALL, NJM ;
BURGEN, ASV ;
HULME, EC ;
STOCKTON, JM ;
ZIGMOND, MJ .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 78 (02) :257-259
[3]  
BITTIGER H, 1981, EXPERIENTIA, V37, P638
[4]   IDENTIFICATION OF AN ACTIVE METABOLITE OF TREMORINE [J].
CHO, AK ;
HASLETT, WL ;
JENDEN, DJ .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1961, 5 (04) :276-&
[5]  
CHO AK, 1962, J PHARMACOL EXP THER, V138, P249
[6]   BINDING-STUDIES WITH [H-3] CIS-METHYLDIOXOLANE IN DIFFERENT TISSUES - UNDER CERTAIN CONDITIONS [H-3] CIS-METHYLDIOXOLANE LABELS PREFERENTIALLY BUT NOT EXCLUSIVELY AGONIST HIGH-AFFINITY STATES OF MUSCARINIC M2-RECEPTORS [J].
CLOSSE, A ;
BITTIGER, H ;
LANGENEGGER, D ;
WANNER, A .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1987, 335 (04) :372-377
[7]   ALKYLATION OF 1-ACYLATED 3-PYRAZOLIDONES AND SYNTHESIS OF 2-SUBSTITUTED 3-PYRAZOLIDONES AND 1-SUBSTITUTED 5-HYDROXYPYRAZOLES [J].
DORN, H ;
ARNDT, D .
JOURNAL FUR PRAKTISCHE CHEMIE, 1971, 313 (01) :115-&
[8]  
DORN H, 1965, Z CHEM, V5, P3377
[9]   MUSCARINIC RECEPTOR SUBTYPES - A CRITIQUE OF THE CURRENT CLASSIFICATION AND A PROPOSAL FOR A WORKING NOMENCLATURE [J].
EGLEN, RM ;
WHITING, RL .
JOURNAL OF AUTONOMIC PHARMACOLOGY, 1986, 6 (04) :323-346
[10]   TREMOR PRODUCED BY DRUGS [J].
EVERETT, GM .
NATURE, 1956, 177 (4522) :1238-1238
123