PHOTOAFFINITY-LABELING OF THE CARDIAC CALCIUM-CHANNEL - (-)-[H-3] AZIDOPINE LABELS A 165-KDA POLYPEPTIDE, AND EVIDENCE AGAINST A [H-3] 1,4-DIHYDROPYRIDINE-ISOTHIOCYANATE BEING A CALCIUM-CHANNEL-SPECIFIC AFFINITY LIGAND

被引:39
作者
FERRY, DR [1 ]
GOLL, A [1 ]
GLOSSMANN, H [1 ]
机构
[1] INST BIOCHEM PHARMAKOL,PETER MAYRSTR 1,A-6020 INNSBRUCK,AUSTRIA
关键词
D O I
10.1042/bj2430127
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:127 / 135
页数:9
相关论文
共 36 条
[1]  
BELLEMANN P, 1981, ARZNEIMITTEL-FORSCH, V31, P2065
[2]  
BOLGER GT, 1983, J PHARMACOL EXP THER, V225, P291
[3]  
BORSOTTO M, 1985, J BIOL CHEM, V260, P4255
[4]  
CAMPBELL KP, 1984, J BIOL CHEM, V259, P5384
[5]   PURIFICATION OF THE CALCIUM-ANTAGONIST RECEPTOR OF THE VOLTAGE-SENSITIVE CALCIUM-CHANNEL FROM SKELETAL-MUSCLE TRANSVERSE TUBULES [J].
CURTIS, BM ;
CATTERALL, WA .
BIOCHEMISTRY, 1984, 23 (10) :2113-2118
[6]   [H-3] NIMODIPINE SPECIFIC BINDING TO CARDIAC MYOCYTES AND SUBCELLULAR-FRACTIONS [J].
DEPOVER, A ;
LEE, SW ;
MATLIB, MA ;
WHITMER, K ;
DAVIS, BA ;
POWELL, T ;
SCHWARTZ, A .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1983, 113 (01) :185-191
[7]   DIHYDROPYRIDINE AND PERIPHERAL TYPE BENZODIAZEPINE BINDING-SITES - SUBCELLULAR-DISTRIBUTION AND MOLECULAR-SIZE DETERMINATION [J].
DOBLE, A ;
BENAVIDES, J ;
FERRIS, O ;
BERTRAND, P ;
MENAGER, J ;
VAUCHER, N ;
BURGEVIN, MC ;
UZAN, A ;
GUEREMY, C ;
LEFUR, G .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 119 (03) :153-167
[8]   THE BINDING OF [H-3]-LABELED NITRENDIPINE TO RECEPTORS FOR CALCIUM-CHANNEL ANTAGONISTS IN THE HEART, CEREBRAL-CORTEX, AND ILEUM OF RATS [J].
EHLERT, FJ ;
ROESKE, WR ;
ITOGA, E ;
YAMAMURA, HI .
LIFE SCIENCES, 1982, 30 (25) :2191-2202
[9]   CALCIUM CHANNELS - EVIDENCE FOR OLIGOMERIC NATURE BY TARGET SIZE ANALYSIS [J].
FERRY, DR ;
GOLL, A ;
GLOSSMANN, H .
EMBO JOURNAL, 1983, 2 (10) :1729-1732
[10]   EVIDENCE FOR MULTIPLE RECEPTOR-SITES WITHIN THE PUTATIVE CALCIUM-CHANNEL [J].
FERRY, DR ;
GLOSSMANN, H .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 321 (01) :80-83