DERIVATIVES OF IMIDAZOLE .3. SYNTHESIS AND PHARMACOLOGICAL ACTIVITIES OF NITRILES AMIDES AND CARBOXYLIC ACID DERIVATIVES OF IMIDAZO(1,2-A)PYRIDINE

被引：32

作者：

ALMIRANTE, L

MUGNAINI, A

RUGARLI, P

GAMBA, A

ZEFELIPPO, E

DETOMA, N

MURMANN, W

机构：

[1] Research Department, Selxi e C, Laboratorio Bioterapico Milanese, Milan

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1969年 / 12卷 / 01期

关键词：

D O I：

10.1021/jm00301a031

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

A number of improved laboratory procedures for the synthesis of imidazol [1,2-a]pyridine derivatives are reported. The resulting compounds, which are structurally related to indole derivatives, have been screened for analgetic, antipyretic, anticonvulsant, and antiinflammatory activity. Phytopharmacological tests have also been performed on the derivatives structurally related to indoleacetic acid. © 1969, American Chemical Society. All rights reserved.

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页码：122 / +

页数：1

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