NOVEL AND FACILE ROUTE TO (+/-)-PHYSOVENINE VIA INTRAMOLECULAR [2+2]CYCLOADDITION REACTION

被引：31
作者：
SHISHIDO, K
AZUMA, T
SHIBUYA, M
机构：
[1] Faculty of Pharmaceutical Sciences, University of Tokushima, Tokushima, 770
来源：
TETRAHEDRON LETTERS | 1990年 / 31卷 / 02期
关键词：
D O I：
10.1016/S0040-4039(00)94375-2
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A formal total synthesis of (±)-physovenine 1 from 2-amino-5-methoxyacetophenone 2 via an intramolecular [2+2]cycloaddition reaction is described. © 1990.
引用
收藏
页码：219 / 220
页数：2
相关论文
共 7 条
[1]   AN APPROACH TO THE BCDE RING OF QUASIMARIN [J].
KRAUS, GA ;
TASCHNER, M ;
SHIMAGAKI, M .
JOURNAL OF ORGANIC CHEMISTRY, 1982, 47 (22) :4271-4274
[2]   CONVERSION OF LACTONES INTO ETHERS [J].
KRAUS, GA ;
FRAZIER, KA ;
ROTH, BD ;
TASCHNER, MJ ;
NEUENSCHWANDER, K .
JOURNAL OF ORGANIC CHEMISTRY, 1981, 46 (11) :2417-2419
[3]  
MARINO JP, 1989, J ORG CHEM, V54, P1784
[4]   CINNOLINES .34. 5-HYDROXY-CINNOLINES,6-HYDROXY-CINNOLINES AND 7-HYDROXY-CINNOLINES AND 5-AMINO-CINNOLINES,6-AMINO-CINNOLINES AND 7-AMINO-CINNOLINES [J].
OSBORN, AR ;
SCHOFIELD, K .
JOURNAL OF THE CHEMICAL SOCIETY, 1955, :2100-2103
[5]   TOTAL SYNTHESES OF (+/-)-PHYSOVENINE AND (+/-)-PHYSOSTIGMINE - AN APPLICATION OF TANDEM ELECTROCYCLIC-[3,3]SIGMATROPIC REACTION OF BENZOCYCLOBUTENES [J].
SHISHIDO, K ;
SHITARA, E ;
KOMATSU, H ;
HIROYA, K ;
FUKUMOTO, K ;
KAMETANI, T .
JOURNAL OF ORGANIC CHEMISTRY, 1986, 51 (15) :3007-3011
[6]   ALKALOID SYNTHESIS VIA THE INTRAMOLECULAR IMIDATE METHYLIDE 1,3-DIPOLAR CYCLO-ADDITION REACTION [J].
SMITH, R ;
LIVINGHOUSE, T .
TETRAHEDRON, 1985, 41 (17) :3559-3568
[7]   INTRAMOLECULAR CYCLO-ADDITION REACTIONS OF KETENES AND KETENIMINIUM SALTS WITH ALKENES [J].
SNIDER, BB .
CHEMICAL REVIEWS, 1988, 88 (05) :793-811
1