A CYCLIC ENKEPHALIN ANALOG WITH HIGH INVITRO OPIATE ACTIVITY

被引：141
作者：
DIMAIO, J [1 ]
SCHILLER, PW [1 ]
机构：
[1] CLIN RES INST MONTREAL, CHEM BIOL & PEPTIDE RES LAB, MONTREAL H2W 1R7, QUEBEC, CANADA
来源：
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES | 1980年 / 77卷 / 12期
关键词：
D O I：
10.1073/pnas.77.12.7162
中图分类号：
Q [生物科学];
学科分类号：
07 ; 0710 ; 09 ;
摘要：
引用
收藏
页码：7162 / 7166
页数：5
相关论文
共 29 条
  • [11] IDENTIFICATION OF 2 RELATED PENTAPEPTIDES FROM BRAIN WITH POTENT OPIATE AGONIST ACTIVITY
    HUGHES, J
    SMITH, TW
    KOSTERLITZ, HW
    FOTHERGILL, LA
    MORGAN, BA
    MORRIS, HR
    [J]. NATURE, 1975, 258 (5536) : 577 - 579
  • [12] PROTON MAGNETIC-RESONANCE STUDIES OF CONFORMATION AND FLEXIBILITY OF ENKEPHALIN PEPTIDES
    JONES, CR
    GIBBONS, WA
    GARSKY, V
    [J]. NATURE, 1976, 262 (5571) : 779 - 782
  • [13] ENDOGENOUS OPIOID PEPTIDES - MULTIPLE AGONISTS AND RECEPTORS
    LORD, JAH
    WATERFIELD, AA
    HUGHES, J
    KOSTERLITZ, HW
    [J]. NATURE, 1977, 267 (5611) : 495 - 499
  • [14] HIGH-AFFINITY ENKEPHALIN-DEGRADING PEPTIDASE IN BRAIN IS INCREASED AFTER MORPHINE
    MALFROY, B
    SWERTS, JP
    GUYON, A
    ROQUES, BP
    SCHWARTZ, JC
    [J]. NATURE, 1978, 276 (5687) : 523 - 526
  • [15] MORGAN BA, 1977, PEPTIDES, P111
  • [16] PASTERNAK GW, 1975, MOL PHARMACOL, V11, P340
  • [17] ACTION OF MORPHINE AND RELATED SUBSTANCES ON CONTRACTION AND ON ACETYLCHOLINE OUTPUT OF COAXIALLY STIMULATED GUINEA-PIG ILEUM
    PATON, WDM
    [J]. BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1957, 12 (01): : 119 - 127
  • [18] D-ALA2-MET-ENKEPHALINAMIDE - POTENT, LONG-LASTING SYNTHETIC PENTAPEPTIDE ANALGESIC
    PERT, CB
    PERT, A
    CHANG, JK
    FONG, BTW
    [J]. SCIENCE, 1976, 194 (4262) : 330 - 332
  • [19] SYNTHESIS, OPIATE RECEPTOR-BINDING AND ANALGESIC ACTIVITY OF ENKEPHALIN ANALOGS
    PLESS, J
    BAUER, W
    CARDINAUX, F
    CLOSSE, A
    HAUSER, D
    HUGUENIN, R
    ROEMER, D
    BUESCHER, HH
    HILL, RC
    [J]. HELVETICA CHIMICA ACTA, 1979, 62 (02) : 398 - 411
  • [20] CONFORMATION OF MET5-ENKEPHALIN DETERMINED BY HIGH-FIELD PMR SPECTROSCOPY
    ROQUES, BP
    GARBAYJAUREGUIBERRY, C
    OBERLIN, R
    ANTEUNIS, M
    LALA, AK
    [J]. NATURE, 1976, 262 (5571) : 778 - 779
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