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- [2] SYNTHESIS OF N-(2,5-[2-C-13]DIMETHYL-1H-PYRROL-1-YL)-6-(4-MORPHOLINYL)-3-PYRIDAZINAMINE HYDROCHLORIDE JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 1985, 22 (12): : 1299 - 1307
- [3] HEMODYNAMIC PROFILE ON N-(2,5-DIMETHYL-1 H-PYRROL-1-YL) 6-(4-MORPHOLINYL)-3-PYRIDAZINAMINE HYDROCHLORIDE IN CONSCIOUS DOGS ARZNEIMITTELFORSCHUNG-DRUG RESEARCH, 1986, 36-1 (01): : 84 - 88
- [5] PHARMACOLOGICAL STUDIES OF N-(2,5-DIMETHYL-1H-PYRROL-1-YL)-6-(4-MORPHOLINYL)-3-PYRIDAZINAMINE HYDROCHLORIDE (MDL-899), A NEW LONG-ACTING ANTIHYPERTENSIVE VASODILATOR ARZNEIMITTELFORSCHUNG-DRUG RESEARCH, 1985, 35-1 (05): : 818 - 826
- [6] Syntheses and pharmacokinetic evaluations of four metabolites of 2-(4-(2-((1H-benzo[d]imidazol-2-yl)thio)ethyl)piperazin-1-yl)-N-(6-methyl-2,4-bis-(methylthio)pyridin-3-yl)acetamide hydrochloride [K-604], an acyl-CoA:cholesterol O-acyltransferase-1 inhibitor BIOORGANIC & MEDICINAL CHEMISTRY, 2020, 28 (11)
- [7] Discovery of Clinical Candidate 2-(4-(2-((1H-Benzo[d]imidazol-2-yl)thio)ethyl)piperazin-1-yl)-N-(6-methyl-2,4-bis(methylthio)pyridin-3-yl)acetannide Hydrochloride [K-604], an Aqueous-Soluble Acyl-CoA:Cholesterol O-Acyltransferase-1 Inhibitor JOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (23) : 10635 - 10650