NONAMINE-CONTAINING BICYCLIC AND TRICYCLIC ANALOGS OF LAVENDUSTIN A AS PROTEIN-TYROSINE KINASE INHIBITORS

被引:0
|
作者
SMYTH, MS
STEFANOVA, I
HARTMANN, F
HORAK, ID
OSHEROV, N
LEVITZKI, A
BURKE, TR
机构
[1] NCI,DCT,DTP,MED CHEM LAB,BETHESDA,MD 20892
[2] NCI,DCBDC,METAB BRANCH,BETHESDA,MD 20892
[3] HEBREW UNIV JERUSALEM,JERUSALEM,ISRAEL
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
引用
收藏
页码:107 / MEDI
相关论文
共 50 条
  • [41] PROTEIN-TYROSINE KINASE INHIBITORS INHIBIT CHEMOTAXIS OF VASCULAR SMOOTH-MUSCLE CELLS
    SHIMOKADO, K
    YOKOTA, T
    UMEZAWA, K
    SASAGURI, T
    OGATA, J
    ARTERIOSCLEROSIS AND THROMBOSIS, 1994, 14 (06): : 973 - 981
  • [42] FLAVONOIDS FROM KOELREUTERIA-HENRYI AND OTHER SOURCES AS PROTEIN-TYROSINE KINASE INHIBITORS
    ABOUSHOER, M
    MA, GE
    LI, XH
    KOONCHANOK, NM
    GEAHLEN, RL
    CHANG, CJ
    JOURNAL OF NATURAL PRODUCTS, 1993, 56 (06): : 967 - 969
  • [43] The role of small molecule Kit protein-tyrosine kinase inhibitors in the treatment of neoplastic disorders
    Roskoski, Robert, Jr.
    PHARMACOLOGICAL RESEARCH, 2018, 133 : 35 - 52
  • [44] Changes and mechanisms of protein-tyrosine kinase and protein-tyrosine phosphatase activities after brain ischemia/reperfusion
    Pei, L
    Li, Y
    Yan, JZ
    Zhang, GY
    Cui, ZC
    Zhu, ZM
    ACTA PHARMACOLOGICA SINICA, 2000, 21 (08) : 715 - 720
  • [45] PROTEIN-TYROSINE PHOSPHATASES AS REGULATORS OF PROTEIN-KINASE ACTIVITY
    SWARUP, G
    RADHA, V
    CURRENT SCIENCE, 1992, 62 (06): : 462 - 469
  • [46] TEC PROTEIN-TYROSINE KINASE DIRECTLY ASSOCIATES WITH LYN PROTEIN-TYROSINE KINASE THROUGH ITS N-TERMINAL UNIQUE DOMAIN
    MANO, H
    SATO, K
    YAZAKI, Y
    HIRAI, H
    ONCOGENE, 1994, 9 (11) : 3205 - 3211
  • [47] Synthesis and SAR of inhibitors of protein kinase CK2: Novel tricyclic quinoline analogs
    Haddach, Mustapha
    Pierre, Fabrice
    Regan, Collin F.
    Borsan, Cosmin
    Michaux, Jerome
    Stefan, Eric
    Kerdoncuff, Pauline
    Schwaebe, Michael K.
    Chua, Peter C.
    Siddiqui-Jain, Adam
    Macalino, Diwata
    Drygin, Denis
    O'Brien, Sean E.
    Rice, William G.
    Ryckman, David M.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (01) : 45 - 48
  • [48] Progress in Research on Protein Tyrosine Kinase Inhibitors Progress in Research on Protein Tyrosine Kinase Inhibitors
    Chen, Yu
    INTERNATIONAL CONFERENCE ON FRONTIERS OF BIOLOGICAL SCIENCES AND ENGINEERING (FBSE 2018), 2019, 2058
  • [49] INHIBITION OF ACROSOME REACTION AND OOCYTE PENETRATION IN NORMOSPERMIC DOMESTIC CATS BY PROTEIN-TYROSINE KINASE INHIBITORS
    PUKAZHENTHI, BS
    WILDT, DE
    OTTINGER, MA
    HOWARD, JG
    BIOLOGY OF REPRODUCTION, 1995, 52 : 58 - 58
  • [50] CYTOSOLIC PROTEIN-TYROSINE KINASE FROM BOVINE PLATELETS
    YAMAMURA, H
    NAKAMURA, S
    THROMBOSIS AND HAEMOSTASIS, 1989, 62 (01) : 462 - 462