A GENERAL-SYNTHESIS OF CHIRAL C-4-ALKYLATED AZETIDIN-2-ONES WHICH ARE OF POTENTIAL USE AS INTERMEDIATES FOR 1BETA-HETEROATOM-SUBSTITUTED CARBAPENEMS

被引：11

作者：

NAGAO, Y

KUMAGAI, T

ABE, T

OCHIAI, M

TAGA, T

MACHIDA, K

INOUE, Y

机构：

[1] KYOTO UNIV,FAC PHARMACEUT SCI,SAKYO KU,KYOTO 606,JAPAN

[2] LEDERLE JAPAN LTD,CHEM & FORMULAT LAB,KASHIWA,SAITAMA 353,JAPAN

来源：

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1987年 / 08期

关键词：

D O I：

10.1039/c39870000602

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

引用

页码：602 / 603

页数：2

共 25 条

[1] 3-(2-alkoxy-1-hydroxyethyl)azetidin-2-ones: Potential intermediates for the synthesis of novel carbapenems
O'Leary, AC
Waldron, CM
Burke, CM
Keaveny, RD
Meegan, MJ
JOURNAL OF CHEMICAL RESEARCH-S, 1998, (02): : 64 - 65A
[2] 4-acetoxy-3-[1-(2-arylamino-1-hydroxy)ethyl]azetidin-2-ones: Intermediates for the synthesis of novel carbapenems
Meegan, MJ
Waldron, CM
Keaveny, RD
Neary, AD
JOURNAL OF CHEMICAL RESEARCH-S, 1997, (05): : 158 - 159
[3] 4-substituted azetidin-2-ones, new building blocks for the synthesis of beta-lactams
Kaluza, Z
Park, SH
SYNLETT, 1996, (09) : 895 - &
[4] N/C-4 substituted azetidin-2-ones: Synthesis and preliminary evaluation as new class of antimicrobial agents
Halve, Arland K.
Bhadauria, Deepti
Dubey, Rakesh
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 17 (02) : 341 - 345
[5] SYNTHESIS AND STEREOCHEMISTRY OF CHIRAL AZETIDIN-2-ONES AND AZETIDIN-2-THIONES .1. SYNTHESIS OF DIASTEREOMERS OF 2-SUBSTITUTED AND 3-SUBSTITUTED N-(ALPHA-METHYLBENZYL)BETA-AMINOPROPIONIC ACIDS
ROMANOVA, NN
TALLO, TG
BUNDEL, YG
ZHURNAL ORGANICHESKOI KHIMII, 1995, 31 (03): : 412 - 415
[6] SYNTHESIS OF BETA-LACTAMS OF HIGH ENANTIOMERIC PURITY BY CHIRAL LIGAND ACCELERATED OSMYLATION OF RACEMIC 4-(2-STYRYL)-AZETIDIN-2-ONES
ANNUNZIATA, R
BENAGLIA, M
CINQUINI, M
COZZI, F
PONZINI, F
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1993, 3 (11) : 2397 - 2402
[7] SYNTHESIS OF 1,3-DIOXIN-4-ONES AND THEIR USE IN SYNTHESIS .18. SYNTHESIS OF AZETIDIN-2-ONES FROM 1,3-DIOXIN-4-ONES VIA 3-HYDROXYCARBOXAMIDES
SAKAKI, J
KOBAYASHI, S
SATO, M
KANEKO, C
CHEMICAL & PHARMACEUTICAL BULLETIN, 1989, 37 (11) : 2952 - 2960
[8] N-ACYL 3-ALKYLIDENYL AZETIDIN-2-ONES AND 3-ALKYL AZETIDIN-2-ONES - A NEW CLASS OF MONOCYCLIC BETA-LACTAM ANTIBACTERIAL AGENTS .2. SYNTHESIS ANDST RUCTURE-ACTIVITY RELATIONSHIPS OF HETEROATOM SUBSTITUTED 3-ISOPROPYLIDENE A ND 3-ISOPROPYL ANALOGS
BRICKNER, SJ
GAIKEMA, JJ
GREENFIELD, LJ
ZURENKO, GE
MANNINEN, PR
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1993, 3 (11) : 2241 - 2246
[9] SYNTHESIS OF A NEW SERIES OF N-SUBSTITUTED-3-[1-ALKYL(ARYL)-4-PIPERIDYL]AZETIDIN-2-ONES AS POSSIBLE MUSCARINIC AGENTS
CIGNARELLA, G
VILLA, S
BARLOCCO, D
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1993, 30 (05) : 1337 - 1340
[10] DESIGN, SYNTHESIS AND ANTIMICROBIAL EVALUATION OF NOVEL 1-(2-(4-FLUORO BENZYLTHIO) PYRIMIDIN-4-YL-AMINO)-4-(SUBSTITUTED PHENYL) AZETIDIN-2-ONES
Goudgaon, N. M.
Reddy, Y. Rohini
INTERNATIONAL JOURNAL OF PHARMACEUTICAL SCIENCES AND RESEARCH, 2015, 6 (03): : 1060 - 1065

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