EXO-SITE AFFINITY LABELING OF C1SBAR, A SUBCOMPONENT OF 1ST COMPONENT OF COMPLEMENT, BY M-[O-(2-CHLORO-5-FLUOROSULFONYLPHENYLUREIDO)PHENOXYBUTOXY]BENZAMIDINE

被引：10

作者：

BING, DH ^{[1
]}

LAURA, R ^{[1
]}

ANDREWS, JM ^{[1
]}

CORY, M ^{[1
]}

机构：

[1] WELLCOME RES LABS,RES TRIANGLE PK,NC 27709

来源：

BIOCHEMISTRY | 1978年 / 17卷 / 26期

关键词：

D O I：

10.1021/bi00619a017

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：5713 / 5718

页数：6

共 33 条

[1]

ANDREWS JM, 1977, J IMMUNOL, V118, P466

[2]

ANDREWS JM, J MED CHEM

[3] IRREVERSIBLE ENZYME INHIBITORS .186. IRREVERSIBLE INHIBITORS OF CLA COMPONENT OF COMPLEMENT DERIVED FROM META-(PHENOXYPROPOXY)BENZAMIDINE BY BRIDGING TO A TERMINAL SULFONYL FLUORIDE [J].

BAKER, BR ;

CORY, M .

JOURNAL OF MEDICINAL CHEMISTRY, 1971, 14 (09) :805-&

[4]

Baker BR, 1967, DESIGN ACTIVE SITE D

[5]

BING DH, 1977, J BIOL CHEM, V252, P8027

[6] NATURE OF ACTIVE SITE OF A SUBUNIT OF FIRST COMPONENT OF HUMAN COMPLEMENT [J].

BING, DH .

BIOCHEMISTRY, 1969, 8 (11) :4503-&

[7]

BING DH, 1974, J IMMUNOL, V113, P584

[8]

BING DH, 1977, CHEM BIOL THROMBIN, P159

[9] IRREVERSIBLE ENZYME INHIBITORS .172. PROTEOLYTIC ENZYMES .16. COVALENT BONDING OF SULFONYL FLUORIDE GROUP TO SERINE OUTSIDE ACTIVE SITE OF ALPHA-CHYMOTRYPSIN BY EXO-TYPE ACTIVE-SITE DIRECTED IRREVERSIBLE INHIBITORS [J].

CARDINAU.R ;

BAKER, BR .

JOURNAL OF MEDICINAL CHEMISTRY, 1970, 13 (03) :467-&

[10] TIME-DEPENDENT INHIBITION OF ENZYMES BY ACTIVE-SITE-DIRECTED REAGENTS A THEORETICAL TREATMENT OF KINETICS OF AFFINITY LABELING [J].

CHILDS, RE ;

BARDSLEY, WG .

JOURNAL OF THEORETICAL BIOLOGY, 1975, 53 (02) :381-394

← 1 2 3 4 →