REGIOSELECTIVE PD-MEDIATED COUPLING BETWEEN 2,6-DICHLOROPURINES AND ORGANOMETALLIC REAGENTS

被引：45

作者：

GUNDERSEN, LL ^{[1
]}

LANGLI, G ^{[1
]}

RISE, F ^{[1
]}

机构：

[1] UNIV OSLO,DEPT CHEM,N-0315 OSLO,NORWAY

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 11期

关键词：

D O I：

10.1016/0040-4039(95)00163-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Selective coupling in the purine 6-position has been achieved, by reacting N-benzylated 2,6-dichloropurines with organotin and organozinc reagents. The positional identity of the products were established from long range HETCOR or nOe NMR experiments.

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页码：1945 / 1948

页数：4

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