STRUCTURE-ACTIVITY-RELATIONSHIPS OF STEROID-HORMONES ON MUSCARINIC RECEPTOR-BINDING

被引:14
作者
KLANGKALYA, B [1 ]
CHAN, A [1 ]
机构
[1] UNIV MISSISSIPPI, MED CTR, DEPT PHARMACOL & TOXICOL, 2500 N STATE ST, JACKSON, MS 39216 USA
关键词
D O I
10.1016/0022-4731(88)90384-6
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:111 / 118
页数:8
相关论文
共 50 条
[21]   MUSCARINIC RECEPTOR-BINDING IS INHIBITED BY QUINACRINE [J].
ODONNELL, KA ;
HOWLETT, AC .
NEUROSCIENCE LETTERS, 1991, 127 (01) :46-48
[22]   MUSCARINIC CHOLINERGIC RECEPTOR-BINDING IN BRAIN [J].
YAMAMURA, HI ;
SNYDER, SH .
FEDERATION PROCEEDINGS, 1974, 33 (03) :467-467
[23]   SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF A NOVEL SERIES OF NONPEPTIDE ANGIOTENSIN-II RECEPTOR-BINDING INHIBITORS SPECIFIC FOR THE AT2 SUBTYPE [J].
BLANKLEY, CJ ;
HODGES, JC ;
KLUTCHKO, SR ;
HIMMELSBACH, RJ ;
CHUCHOLOWSKI, A ;
CONNOLLY, CJ ;
NEERGAARD, SJ ;
VANNIEUWENHZE, MS ;
SEBASTIAN, A ;
QUIN, J ;
ESSENBURG, AD ;
COHEN, DM .
JOURNAL OF MEDICINAL CHEMISTRY, 1991, 34 (11) :3248-3260
[24]   SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF NOVEL AMIDINE DERIVATIVES AS MUSCARINIC RECEPTOR SUBTYPE-SELECTIVE AGONISTS [J].
OJO, B ;
DUNBAR, PG ;
DURANT, GJ ;
HUZL, JJ ;
ELASSADI, AA ;
PERIYASAMY, S ;
NGUR, DO ;
HOSS, WP ;
MESSER, WS .
LIFE SCIENCES, 1995, 56 (11-12) :1005-1005
[25]   GAP JUNCTION MODULATION IN RAT UTERUS .3. STRUCTURE-ACTIVITY-RELATIONSHIPS OF ESTROGEN RECEPTOR-BINDING LIGANDS ON MYOMETRIAL AND SEROSAL CELLS [J].
BURGHARDT, RC ;
GADDYKURTEN, D ;
BURGHARDT, RL ;
KURTEN, RC ;
MITCHELL, PA .
BIOLOGY OF REPRODUCTION, 1987, 36 (03) :741-751
[26]   DIPYRAZOLO[5,4-B-3',4'-D]PYRIDINES - SYNTHESIS, INHIBITION OF BENZODIAZEPINE RECEPTOR-BINDING AND STRUCTURE-ACTIVITY-RELATIONSHIPS [J].
MELANI, F ;
CECCHI, L ;
COLOTTA, V ;
FILACCHIONI, G ;
MARTINI, C ;
GIANNACCINI, G ;
LUCACCHINI, A .
FARMACO, 1989, 44 (06) :585-594
[27]   INVITRO BINDING OF STEROID-HORMONES BY NATURAL AND PURIFIED FIBERS [J].
SHULTZ, TD ;
HOWIE, BJ .
FEDERATION PROCEEDINGS, 1986, 45 (03) :349-349
[28]   QUANTITATIVE STRUCTURE-ACTIVITY-RELATIONSHIPS COMPARATIVE MOLECULAR-FIELD ANALYSIS (QSAR/COMFA) FOR RECEPTOR-BINDING PROPERTIES OF HALOGENATED ESTRADIOL DERIVATIVES [J].
GANTCHEV, TG ;
ALI, H ;
VANLIER, JE .
JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (24) :4164-4176
[29]   EFFECTS OF HYPERTHYROIDISM ON BINDING-PROTEINS FOR STEROID-HORMONES [J].
CARON, P ;
BENNET, A ;
BAROUSSE, C ;
NISULA, BC ;
LOUVET, JP .
CLINICAL ENDOCRINOLOGY, 1989, 31 (02) :219-224
[30]   STEROID-HORMONES AND BINDING-PROTEINS IN SALIVARY TISSUE [J].
WALDEN, WE ;
WITTLIFF, JL .
JOURNAL OF DENTAL RESEARCH, 1983, 62 :266-266