SYNTHESIS AND ANTIVIRAL ACTIVITY OF 3-SUBSTITUTED IMIDAZO[1,2-A]PYRIDINES

被引：85
|
作者：
ELHAKMAOUI, A
GUEIFFIER, A
MILHAVET, JC
BLACHE, Y
CHAPAT, JP
CHAVIGNON, O
TEULADE, JC
SNOECK, R
ANDREI, G
DECLERCQ, E
机构：
[1] LAB CHIM ORGAN PHARMACEUT,CNRS,URA 1111,F-34060 MONTPELLIER,FRANCE
[2] UNIV AUVERGNE,FAC PHARM,DEPT CHIM STRUCT & PHARMACOCHIM,F-63001 CLERMONT FERRAND,FRANCE
[3] KATHOLIEKE UNIV LEUVEN,REGA INST MED RES,B-3000 LOUVAIN,BELGIUM
来源：
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1994年 / 4卷 / 16期
关键词：
D O I：
10.1016/S0960-894X(01)80538-2
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
A series of 3-substituted imidazo[1,2-a]pyridines was synthesized as potential antiviral agents. Compound 10b and, to a lesser extent, 10c showed activity against both TK+ and TK- strains of varicella-zoster virus.
引用
收藏
页码：1937 / 1940
页数：4
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