MODELING OF STRUCTURE OF HUMAN IMMUNODEFICIENCY VIRUS-1 PROTEASE WITH SUBSTRATE BASED ON CRYSTAL-STRUCTURE OF ROUS-SARCOMA VIRUS PROTEASE

被引:0
|
作者
WEBER, IT
机构
关键词
D O I
暂无
中图分类号
Q5 [生物化学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:727 / 741
页数:15
相关论文
共 50 条
  • [1] MUTATIONAL ANALYSIS OF THE SUBSTRATE-BINDING POCKETS OF THE ROUS-SARCOMA VIRUS AND HUMAN IMMUNODEFICIENCY VIRUS-1 PROTEASES
    CAMERON, CE
    RIDKY, TW
    SHULENIN, S
    LEIS, J
    WEBER, IT
    COPELAND, T
    WLODAWER, A
    BURSTEIN, H
    BIZUBBENDER, D
    SKALKA, AM
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1994, 269 (15) : 11170 - 11177
  • [2] DOMAIN COMMUNICATION IN THE DYNAMIC STRUCTURE OF HUMAN IMMUNODEFICIENCY VIRUS-1 PROTEASE
    HARTE, WE
    SWAMINATHAN, S
    MANSURI, MM
    MARTIN, JC
    ROSENBERG, IE
    BEVERIDGE, DL
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1990, 87 (22) : 8864 - 8868
  • [3] Structure based prediction of binding affinity of human immunodeficiency virus-1 protease inhibitors
    Kulkarni, SS
    Kulkarni, VM
    JOURNAL OF CHEMICAL INFORMATION AND COMPUTER SCIENCES, 1999, 39 (06): : 1128 - 1140
  • [4] Structure Based Prediction of Binding Affinity of Human Immunodeficiency Virus-1 Protease Inhibitors
    Kulkarni, Santosh S.
    Kulkarni, Vithal M.
    Journal of Chemical Information and Computer Sciences, 39 (06): : 1128 - 1140
  • [5] MUTATIONS THAT ALTER THE ACTIVITY OF THE ROUS-SARCOMA VIRUS PROTEASE
    GRINDE, B
    CAMERON, CE
    LEIS, J
    WEBER, IT
    WLODAWER, A
    BURSTEIN, H
    BIZUB, D
    SKALKA, AM
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1992, 267 (14) : 9481 - 9490
  • [6] ANALYSIS OF SUBSTRATE INTERACTIONS OF THE ROUS-SARCOMA VIRUS WILD-TYPE AND MUTANT PROTEASES AND HUMAN IMMUNODEFICIENCY VIRUS-1 PROTEASE USING A SET OF SYSTEMATICALLY ALTERED PEPTIDE-SUBSTRATES
    GRINDE, B
    CAMERON, CE
    LEIS, J
    WEBER, IT
    WLODAWER, A
    BURSTEIN, H
    SKALKA, AM
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1992, 267 (14) : 9491 - 9498
  • [7] INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS-1 PROTEASE
    TYAGI, SC
    BIOCHEMISTRY AND CELL BIOLOGY-BIOCHIMIE ET BIOLOGIE CELLULAIRE, 1992, 70 (05): : 309 - 315
  • [8] RIBONUCLEASE-A AS A SUBSTRATE OF THE PROTEASE FROM HUMAN IMMUNODEFICIENCY VIRUS-1
    HUI, JO
    TOMASSELLI, AG
    ZURCHERNEELY, HA
    HEINRIKSON, RL
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1990, 265 (34) : 21386 - 21389
  • [9] STRUCTURE-BASED DESIGN OF NONPEPTIDE INHIBITORS SPECIFIC FOR THE HUMAN IMMUNODEFICIENCY VIRUS-1 PROTEASE
    DESJARLAIS, RL
    SEIBEL, GL
    KUNTZ, ID
    FURTH, PS
    ALVAREZ, JC
    DEMONTELLANO, PRO
    DECAMP, DL
    BABE, LM
    CRAIK, CS
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1990, 87 (17) : 6644 - 6648
  • [10] STRUCTURE-ASSISTED DESIGN OF NONPEPTIDE HUMAN IMMUNODEFICIENCY VIRUS-1 PROTEASE INHIBITORS
    ROSE, JR
    CRAIK, CS
    AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE, 1994, 150 (06) : S176 - S182