A NEW APPROACH TO THE SYNTHESIS OF BETA-FLUOROPYRROLE DERIVATIVES

被引：25

作者：

QIU, ZM ^{[1
]}

BURTON, DJ ^{[1
]}

机构：

[1] UNIV IOWA,DEPT CHEM,IOWA CITY,IA 52242

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 25期

基金：

美国国家科学基金会;

关键词：

D O I：

10.1016/S0040-4039(00)73343-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

beta-Fluoropyrrole derivatives are synthesized in high yields by the reaction of alpha,alpha-difluoro-gamma-iodo-gamma-(electron-withdrawing-group)-substituted ketones and ammonium hydroxide at room temperature; providing a new, simple, and efficient method for the synthesis of beta-fluorinated pyrrole rings. A possible mechanism is proposed.

引用

页码：4319 / 4322

页数：4

共 50 条

[21] NEW APPROACH TO THE SYNTHESIS OF DEOXYNUCLEOSIDE-PHOSPHORAMIDITE DERIVATIVES
TANAKA, T
TAMATSUKURI, S
IKEHARA, M
TETRAHEDRON LETTERS, 1986, 27 (02) : 199 - 202
[22] A NEW APPROACH FOR THE SYNTHESIS OF SOME BENZOXAZINONE AND QUINAZOLINONE DERIVATIVES
SOLIMAN, FM
ISLAM, IE
KASSAB, RR
SOUKA, LM
ELKADY, MY
REVUE ROUMAINE DE CHIMIE, 1994, 39 (04) : 405 - 411
[23] NEW APPROACH TO SYNTHESIS OF DIBENZO[A,D]CYCLOHEPTATRIENE DERIVATIVES
BROVCHENKO, VG
BICHEROV, AV
KUZNETSOV, EV
ZHURNAL ORGANICHESKOI KHIMII, 1984, 20 (01): : 224 - 225
[24] New approach to synthesis of 4-arylcoumarin derivatives
Bardasov, Ivan N.
Alekseeva, Anastasiya U.
Ershov, Oleg V.
Surazhskaya, Marina D.
Churakov, Andrei V.
Grishanov, Dmitry A.
TETRAHEDRON LETTERS, 2015, 56 (44) : 6145 - 6148
[25] New Approach to the Synthesis of Biologically Active Derivatives of Pyranocoumarins
Inyutina, A. K.
Fatykhov, R. F.
Khalymbadzha, I. A.
Sharapov, A. D.
Bobkina, M., V
Chupakhin, O. N.
PROCEEDINGS OF THE II INTERNATIONAL CONFERENCE: MODERN SYNTHETIC METHODOLOGIES FOR CREATING DRUGS AND FUNCTIONAL MATERIALS (MOSM2018), 2019, 2063
[26] New approach to the synthesis of lysophosphatidylcholines and related derivatives.
Hajdu, J
Bibak, N
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2003, 226 : U103 - U103
[27] A NEW APPROACH FOR THE SYNTHESIS OF SOME PYRIDINE AND PYRIDONE DERIVATIVES
HISHMAT, OH
ZOHAIR, MMY
MIKY, JAA
ZEITSCHRIFT FUR NATURFORSCHUNG SECTION B-A JOURNAL OF CHEMICAL SCIENCES, 1983, 38 (12): : 1690 - 1694
[28] A new approach to the stereoselective synthesis of beta-methylchalcones
Elmorsy, SS
Khalil, AGM
Girges, MM
Salama, TA
JOURNAL OF CHEMICAL RESEARCH-S, 1997, (07): : 232 - &
[29] ACTIVATED NITRILES IN HETEROCYCLIC SYNTHESIS - A NEW APPROACH FOR THE SYNTHESIS OF PYRAN DERIVATIVES
IBRAHIM, NS
HETEROCYCLES, 1986, 24 (04) : 935 - 938
[30] A NEW APPROACH TO THE SYNTHESIS OF 2-BETA AND 3-BETA-HYDROXYGIBBERELLINS
WILLIS, CL
TETRAHEDRON LETTERS, 1987, 28 (52) : 6705 - 6708

← 1 2 3 4 5 →