METHIODIDE APPROACH TO THE SYNTHESIS OF 3-[2-(DIMETHYLAMINO)ETHYL]-5-[(1,1-DIOXO-5-METHYL-1,2,5-THIADIAZOLIDIN-2-YL)METHYL]-1H-INDOLE AND ANALOGS

被引：18

作者：

CASTRO, JL

MATASSA, VG

机构：

[1] Medicinal Chemistry Department, Merck Sharp md Dohme Research Laboratories, Neuroscience Research Centre, Harlow, Essex CM20 2QR, Terlings Park, Eastwick Road

来源：

TETRAHEDRON LETTERS | 1993年 / 34卷 / 29期

关键词：

D O I：

10.1016/S0040-4039(00)60662-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Tryptamines 1, 2 and 3 have been synthesised in a convergent and efficient manner by reaction of a novel methiodide 4c with the anions of the cyclic sulphamides 5, 6 and 7 as the key step.

引用

页码：4705 / 4708

页数：4

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