SYNTHESIS OF OPTICALLY-ACTIVE A-RING FRAGMENTS OF TAXOL VIA ELECTROPHILIC RING-CLOSURE OF AN EPOXY-ALLYLSILANE

被引：18

作者：

PETTERSSON, L ^{[1
]}

MAGNUSSON, G ^{[1
]}

FREJD, T ^{[1
]}

机构：

[1] UNIV LUND,LUND INST TECHNOL,CTR CHEM,S-22100 LUND,SWEDEN

来源：

ACTA CHEMICA SCANDINAVICA | 1993年 / 47卷 / 02期

关键词：

D O I：

10.3891/acta.chem.scand.47-0196

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

The optically active A-ring fragment 3 (and related derivatives) of taxol (1) has been synthesized via electrophilic ring closure of an optically active epoxy-allylsilane, prepared from L-arabinose.

引用

页码：196 / 207

页数：12

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