共 21 条
[2]
[2',5'-BIS-O-(TERT-BUTYLDIMETHYLSILYL)]-3'-SPIRO-5''-(4''-AMINO-1'',2''-OXATHIOLE-2'',2''-DIOXIDE) (TSAO) DERIVATIVES OF PURINE AND PYRIMIDINE NUCLEOSIDES AS POTENT AND SELECTIVE INHIBITORS OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1
[J].
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY,
1992, 36 (05)
:1073-1080
[3]
2',5'-BIS-O-(TERT-BUTYLDIMETHYLSILYL)-3'-SPIRO-5''-(4''-AMINO-1',2''-OXATHIOLE-2'',2''-DIOXIDE)PYRIMIDINE (TSAO) NUCLEOSIDE ANALOGS - HIGHLY SELECTIVE INHIBITORS OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 THAT ARE TARGETED AT THE VIRAL REVERSE-TRANSCRIPTASE
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1992, 89 (10)
:4392-4396
[4]
BALZARINI J, 1992, 3RD P INT S CHEM SYN
[5]
3'-SPIRO NUCLEOSIDES, A NEW CLASS OF SPECIFIC HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 INHIBITORS - SYNTHESIS AND ANTIVIRAL ACTIVITY OF [2',5'-BIS-O-(TERT-BUTYLDIMETHYLSILYL)-BETA-D-XYLO AND RIBOFURANOSE]-3'-SPIRO-5''-[4''-AMINO-1'',2''-OXATHIOLE 2'',2''-DIOXIDE] (TSAO) PYRIMIDINE NUCLEOSIDES
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1992, 35 (15)
:2721-2727
[6]
DOSHI KJ, 1989, DRUG METAB DISPOS, V17, P590
[7]
EISEMAN JL, 1988, FASEB J, V2, pA913
[9]
DETERMINATION OF 2',3'-DIDEOXYADENOSINE, 2',3'-DIDEOXYINOSINE AND 2',3'-DIDEOXYCYTIDINE IN BIOLOGICAL SAMPLES
[J].
JOURNAL OF CHROMATOGRAPHY-BIOMEDICAL APPLICATIONS,
1988, 431 (01)
:184-191
[10]
KELLEY JA, 1987, DRUG METAB DISPOS, V15, P595