THE INTERACTION OF PHENYLALKYLAMINE CALCIUM-CHANNEL BLOCKERS WITH THE 1,4-DIHYDROPYRIDINE BINDING-SITE

被引:15
|
作者
ZOBRIST, RH
GIACOMINI, KM
NELSON, WL
GIACOMINI, JC
机构
[1] STANFORD UNIV, VET ADM MED CTR, MED CTR, DIV CARDIOL, STANFORD, CA 94305 USA
[2] UNIV CALIF SAN FRANCISCO, SCH PHARM, SAN FRANCISCO, CA 94143 USA
[3] UNIV CALIF SAN FRANCISCO, SCH MED, SAN FRANCISCO, CA 94143 USA
[4] UNIV WASHINGTON, SCH PHARM, SEATTLE, WA 98198 USA
关键词
D O I
10.1016/S0022-2828(86)80010-4
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:963 / 974
页数:12
相关论文
共 50 条
  • [31] Brain pharmacokinetics and in vivo receptor binding of 1,4-dihydropyridine calcium channel antagonists
    Uchida, S
    Yamada, S
    Nagai, K
    Deguchi, Y
    Kimura, Y
    LIFE SCIENCES, 1997, 61 (21) : 2083 - 2090
  • [32] EFFECT OF INORGANIC CALCIUM-CHANNEL BLOCKERS ON DIHYDROPYRIDINE BINDING TO CARDIAC SARCOLEMMA
    SCHILLING, WP
    ZAHER, MC
    RAMPE, D
    MOLECULAR PHARMACOLOGY, 1990, 37 (01) : 80 - 89
  • [33] Obtaining antibodies to 1,4-Dihydropyridine calcium channel antagonists
    A. A. Burkin
    M. A. Burkin
    Applied Biochemistry and Microbiology, 2008, 44 : 323 - 327
  • [34] QSAR STUDY ON 1,4-DIHYDROPYRIDINE AS CALCIUM CHANNEL ANTAGONISTS
    Singh, J.
    Shaik, B.
    Shukla, S. K.
    Sharma, M.
    Singh, S.
    Agrawal, V. K.
    OXIDATION COMMUNICATIONS, 2013, 36 (03): : 761 - 777
  • [35] Obtaining antibodies to 1,4-dihydropyridine calcium channel antagonists
    Burkin, A. A.
    Burkin, M. A.
    APPLIED BIOCHEMISTRY AND MICROBIOLOGY, 2008, 44 (03) : 323 - 327
  • [36] QSAR Analysis of 1,4-Dihydropyridine Calcium Channel Antogonists
    Kahraman, Pinar
    Turkay, Metin
    17TH EUROPEAN SYMPOSIUM ON COMPUTER AIDED PROCESS ENGINEERING, 2007, 24 : 977 - 982
  • [37] PROISCHEMIC COMPLICATIONS OF DIHYDROPYRIDINE CALCIUM-CHANNEL BLOCKERS
    WATERS, D
    CIRCULATION, 1991, 84 (06) : 2598 - 2600
  • [39] MOLECULAR-LEVEL MODEL FOR THE AGONIST ANTAGONIST SELECTIVITY OF THE 1,4-DIHYDROPYRIDINE CALCIUM-CHANNEL RECEPTOR
    LANGS, DA
    KWON, YW
    STRONG, PD
    TRIGGLE, DJ
    JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 1991, 5 (02) : 95 - 106
  • [40] PURIFICATION AND CHARACTERIZATION OF THE PUTATIVE CALCIUM-CHANNEL (1,4-DIHYDROPYRIDINE RECEPTOR) FROM SKELETAL-MUSCLE
    NAKAYAMA, N
    KIRLEY, TL
    VAGHY, PL
    SCHWARTZ, A
    CIRCULATION, 1986, 74 (04) : 81 - 81