INHIBITION OF ACETYL-COENZYME A CARBOXYLASE BY THE NOVEL GRASS-SELECTIVE HERBICIDE 3-(2,4-DICHLOROPHENYL)-PERHYDROINDOLIZINE-2,4-DIONE

被引：17

作者：

BABCZINSKI, P ^{[1
]}

FISCHER, R ^{[1
]}

机构：

[1] BAYER AG,PFLANZENSCHUTZZENTRUM MONHEIM,CHEM RES,W-5090 LEVERKUSEN,GERMANY

来源：

PESTICIDE SCIENCE | 1991年 / 33卷 / 04期

关键词：

D O I：

10.1002/ps.2780330408

中图分类号：

S3 [农学（农艺学）];

学科分类号：

0901 ;

摘要：

The novel herbicidal compound 3-(2,4-dichlorophenyl)-perhydroindolizine-2,4-dione which is active as a pre- and post-emergence grass-selective herbicide is a new type of inhibitor of plant acetyl-coenzyme A carboxylase (ACCase; E. C. 6.4.1.2). This has been demonstrated by in-vitro experiments using isolated corn enzyme. Besides an I50 value of 4.7-mu-M under the assay conditions used, a mixed-type inhibitory activity on the enzyme is established. The compound is inactive on rat liver ACCase enzyme and shows decreased activity (pI50 less than 3.0) on the spinach enzyme.

引用

页码：455 / 466

页数：12

共 22 条

[1] INHIBITION OF PLANT ACETYL-COENZYME-A CARBOXYLASE BY THE NOVEL GRASS-SELECTIVE HERBICIDE 3-(2,4-DICHLOROPHENYL)-1-AZA-BICYCLO-(4,3,01,5)-2,4-DIONE
BABCZINSKI, P
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[2] INHIBITION OF ACETYL-COENZYME-A CARBOXYLASE BY 2 CLASSES OF GRASS-SELECTIVE HERBICIDES
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