DIVERSION OF PROSTAGLANDIN ENDOPEROXIDE METABOLISM BY SELECTIVE-INHIBITION OF THROMBOXANE A2 BIOSYNTHESIS IN LUNG, SPLEEN OR PLATELETS

被引:134
|
作者
NIJKAMP, FP
MONCADA, S
WHITE, HL
VANE, JR
机构
[1] WELLCOME RES LABS,BECKENHAM BR3 3BS,KENT,ENGLAND
[2] WELLCOME RES LABS,RES TRIANGLE PK,NC 27709
关键词
D O I
10.1016/0014-2999(77)90104-2
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:179 / 186
页数:8
相关论文
共 50 条
  • [31] INHIBITION OF PGE1-STIMULATED CAMP ACCUMULATION IN HUMAN PLATELETS BY THROMBOXANE A2
    MILLER, OV
    JOHNSON, RA
    GORMAN, RR
    PROSTAGLANDINS, 1977, 13 (04): : 599 - 609
  • [32] THROMBOXANE A2 - KEY REGULATOR OF PROSTAGLANDIN BIOSYNTHESIS AND OF INTERACTIONS BETWEEN PROSTAGLANDINS, CALCIUM AND CYCLIC NUCLEOTIDES
    HORROBIN, DF
    MANKU, MS
    KARMALI, RA
    OKA, M
    ALLY, AI
    MORGAN, RO
    KARMAZYN, M
    CUNNANE, SC
    MEDICAL HYPOTHESES, 1978, 4 (02) : 178 - 186
  • [33] Effect of thromboxane A2 inhibition and antagonism on prostaglandin and leukotriene synthesis in glomerular immune injury
    Lianos, EA
    Bresnahan, BA
    JOURNAL OF LABORATORY AND CLINICAL MEDICINE, 1999, 134 (05): : 478 - 482
  • [34] SELECTIVE-INHIBITION OF RENAL THROMBOXANE BIOSYNTHESIS INCREASED SODIUM-EXCRETION RATE IN NORMAL AND SALINE-LOADED RATS
    PAPANICOLAOU, N
    GKIKA, EL
    GKIKAS, G
    BARIETY, J
    CLINICAL SCIENCE, 1985, 68 (01) : 79 - 82
  • [35] DIFFERENTIAL-EFFECTS OF OKY-046, A SELECTIVE THROMBOXANE (TX)-SYNTHASE INHIBITOR, ON PLATELET AND RENAL PROSTAGLANDIN (PG) ENDOPEROXIDE METABOLISM
    PATRIGNANI, P
    CATELLA, F
    FILABOZZI, P
    PUGLIESE, F
    PIERUCCI, A
    SIMONETTI, B
    FORNI, L
    SEGNI, M
    PATRONO, C
    CLINICAL RESEARCH, 1984, 32 (02): : A246 - A246
  • [36] SYNTHESIS OF A NEW PROSTAGLANDIN ENDOPEROXIDE (PGH2) ANALOG AND ITS FUNCTION AS AN INHIBITOR OF THE BIOSYNTHESIS OF THROMBOXANE-A2(TBXA2)
    COREY, EJ
    NIWA, H
    BLOOM, M
    RAMWELL, PW
    TETRAHEDRON LETTERS, 1979, (08) : 671 - 674
  • [37] STUDIES OF THE REACTIONS OF PGH2, THE ENDOPEROXIDE INTERMEDIATE IN PROSTAGLANDIN AND THROMBOXANE BIOSYNTHESIS, BY H-1-NMR AT 500 MHZ
    ANDERSEN, NH
    WILSON, CH
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1983, 185 (MAR): : 267 - ORGN
  • [38] DUAL INHIBITION OF THROMBOXANE-A2 SYNTHESIS AND THROMBOXANE-A2 PROSTAGLANDIN ENDOPEROXIDE RECEPTORS BY RIDOGREL - ANTITHROMBOTIC EFFECT INVIVO IN RAT MESENTERIC-ARTERIES
    BOURGAIN, RH
    ANDRIES, R
    DECUYPER, K
    DECLERCK, F
    JOURNAL OF LIPID MEDIATORS, 1991, 3 (01): : 3 - 11
  • [39] PROSTACYCLIN AND THROMBOXANE A2 BIOSYNTHESIS CAPACITIES OF HEART, ARTERIES AND PLATELETS AT VARIOUS STAGES OF EXPERIMENTAL ATHEROSCLEROSIS IN RABBITS
    GRYGLEWSKI, RJ
    DEMBINSKAKIEC, A
    ZMUDA, A
    GRYGLEWSKA, T
    ATHEROSCLEROSIS, 1978, 31 (04) : 385 - 394
  • [40] The role of inhibition of nitric oxide synthesis in the aggregation of platelets due to the stimulated production of thromboxane A2
    Banerjee, Debipriya
    Mazumder, Sahana
    Sinha, Asru K.
    BLOOD COAGULATION & FIBRINOLYSIS, 2014, 25 (06) : 585 - 591