NEW 2-IODO SUBSTITUTED DERIVATIVES OF IDAZOXAN WITH HIGH-AFFINITY FOR MAMMALIAN ALPHA(2)-ADRENOCEPTORS

被引:0
作者
HUDSON, AL
NUTT, DJ
LEWIS, JW
MALLARD, NJ
CHAPLEO, CB
机构
[1] SCH MED SCI,DEPT PHARMACOL,PSYCHOPHARMACOL UNIT,BRISTOL BS8 1TD,ENGLAND
[2] UNIV WALES COLL MED,CARDIFF CLIN TRIALS LTD,CARDIFF CF4 4XN,S GLAM,WALES
[3] RECKITT & COLMAN LTD,KINGSTON HULL HU8 7DS,N HUMBERSIDE,ENGLAND
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:P24 / P24
页数:1
相关论文
共 50 条
[21]   Synthesis of new pyridazinone derivatives and their affinity towards α1-α2-adrenoceptors [J].
Corsano, S ;
Strappaghetti, G ;
Barbaro, R ;
Giannaccini, G ;
Betti, L ;
Lucacchini, A .
BIOORGANIC & MEDICINAL CHEMISTRY, 1999, 7 (05) :933-941
[22]   NEW FLUORINE-SUBSTITUTED ANALOG OF ETICLOPRIDE WITH HIGH-AFFINITY TOWARD DOPAMINE D2 RECEPTORS [J].
WATANABE, K ;
FUKUMURA, T ;
SASAKI, S ;
MAEDA, M ;
TAKEHARA, S .
CHEMICAL & PHARMACEUTICAL BULLETIN, 1991, 39 (12) :3211-3214
[23]   [H-3] RS-15385-197, A SELECTIVE AND HIGH-AFFINITY RADIOLIGAND FOR ALPHA-2-ADRENOCEPTORS - IMPLICATIONS FOR RECEPTOR CLASSIFICATION [J].
MACKINNON, AC ;
KILPATRICK, AT ;
KENNY, BA ;
SPEDDING, M ;
BROWN, CM .
BRITISH JOURNAL OF PHARMACOLOGY, 1992, 106 (04) :1011-1018
[24]   RECOMBINANT ALPHA(2)M RECEPTOR-BINDING DOMAIN BINDS TO THE ALPHA(2)M RECEPTOR WITH HIGH-AFFINITY [J].
HOLTET, TL ;
NIELSEN, KL ;
ETZERODT, M ;
MOESTRUP, SK ;
GLIEMANN, J ;
SOTTRUPJENSEN, L ;
THOGERSEN, HC .
BIOLOGY OF ALPHA2-MACROGLOBULIN, ITS RECEPTOR, AND RELATED PROTEINS, 1994, 737 :480-482
[25]   NEW INSIGHTS INTO THE STRUCTURE OF HIGH-AFFINITY INTERLEUKIN-2 RECEPTORS [J].
GREENE, WC ;
WANO, Y ;
DUKOVICH, M .
RECENT PROGRESS IN HORMONE RESEARCH, 1988, 44 :141-155
[26]   [I-125]-HEAT, A SELECTIVE, HIGH-AFFINITY, HIGH SPECIFIC ACTIVITY LIGAND FOR ALPHA-1-ADRENOCEPTORS [J].
GLOSSMANN, H ;
LUBBECKE, F ;
BELLEMANN, P .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1981, 318 (01) :1-9
[27]   Immunosuppressive and anticancer effect of a mammalian ribonuclease that targets high-affinity interleukin-2-receptors [J].
Yamamura, T ;
Ueda, M ;
Psarras, K ;
Suwa, T ;
Watanaabe, Y ;
Kameyama, N ;
Tanabe, M ;
Imamura, H ;
Kitajima, M .
EUROPEAN JOURNAL OF SURGERY, 2002, 168 (01) :49-54
[28]   [H-3] IDAZOXAN BINDING AT NON-ALPHA-2-ADRENOCEPTORS IN RABBIT ADIPOCYTE MEMBRANES [J].
LANGIN, D ;
LAFONTAN, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1989, 159 (02) :199-203
[29]   SYNTHESIS AND CHARACTERIZATION OF A HIGH-AFFINITY RADIOIODINATED PROBE FOR THE ALPHA-2-ADRENERGIC RECEPTOR [J].
LANIER, SM ;
HESS, HJ ;
GRODSKI, A ;
GRAHAM, RM ;
HOMCY, CJ .
MOLECULAR PHARMACOLOGY, 1986, 29 (03) :219-227
[30]   DENSITY OF ALPHA-2A ADRENOCEPTORS AND G(I) PROTEINS IN THE HUMAN BRAIN - RATIO OF HIGH-AFFINITY AGONIST SITES TO ANTAGONIST SITES AND EFFECT OF AGE [J].
SASTRE, M ;
GARCIASEVILLA, JA .
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1994, 269 (03) :1062-1072