BLOCKADE OF MUSCARINIC RECEPTORS BY ALKYLATING AGONIST ANALOGS

被引:5
作者
HULME, EC [1 ]
SPALDING, TA [1 ]
CURTIS, CAM [1 ]
BIRDSALL, NJM [1 ]
CORRIE, JET [1 ]
机构
[1] NATL INST MED RES,DIV PHYS BIOCHEM,LONDON NW7 1AA,ENGLAND
关键词
D O I
10.1042/bst0180440
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:440 / 441
页数:2
相关论文
共 6 条
[1]  
BAKER SP, 1986, MOL PHARMACOL, V30, P411
[2]  
CURTIS CAM, 1989, J BIOL CHEM, V264, P489
[3]   MUSCARINIC RECEPTOR SUBTYPES [J].
HULME, EC ;
BIRDSALL, NJM ;
BUCKLEY, NJ .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1990, 30 :633-673
[4]  
HULME EC, 1989, TRENDS PHARMACOL SCI, V10, P22
[5]   IRREVERSIBLE BINDING OF ACETYLCHOLINE MUSTARD TO MUSCARINIC RECEPTORS IN INTESTINAL SMOOTH-MUSCLE OF GUINEA-PIG [J].
ROBINSON, DA ;
TAYLOR, JG ;
YOUNG, JM .
BRITISH JOURNAL OF PHARMACOLOGY, 1975, 53 (03) :363-370
[6]   THE STRUCTURE AND PROPERTIES OF THE PURIFIED MUSCARINIC ACETYLCHOLINE-RECEPTOR FROM RAT FOREBRAIN [J].
WHEATLEY, M ;
BIRDSALL, NJM ;
CURTIS, C ;
EVELEIGH, P ;
PEDDER, EK ;
POYNER, D ;
STOCKTON, JM ;
HULME, EC .
BIOCHEMICAL SOCIETY TRANSACTIONS, 1987, 15 (01) :113-116