SYNTHESIS OF OPTICALLY-ACTIVE 1-FLUOROALKYL BENZENES

被引：6

作者：

FRITZLANGHALS, E

机构：

[1] Consortium für Elektrochemische Industrie GmbH, Central Research Company, Wacker-Chemie GmbH, D-81379 München

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 12期

关键词：

D O I：

10.1016/S0040-4039(00)73178-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A simple synthesis of optically active 1-fluoroalkyl benzenes bearing electron withdrawing substituents is developed. Optically active 1-hydroxyalkyl benzenes are converted into the methanesulfonates and subsequently converted into the optically active 1-fluoroalkyl benzenes 1 by use of the fluorinating agent cesium fluoride/N-methyl-formamide.

引用

页码：1851 / 1854

页数：4

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