TOTAL SYNTHESIS OF THE SPIROKETAL MACROLIDE (+) MILBEMYCIN ALPHA(1)

被引：8

作者：

LEY, SV ^{[1
]}

MADIN, A ^{[1
]}

MONCK, NJT ^{[1
]}

机构：

[1] UNIV LONDON IMPERIAL COLL SCI TECHNOL & MED,LONDON SW7 2AY,ENGLAND

来源：

TETRAHEDRON LETTERS | 1993年 / 34卷 / 46期

关键词：

D O I：

10.1016/S0040-4039(00)60158-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The total synthesis of the antiparasitic spiroketal macrolide (+) milbemycin alpha1 is reported, following Julia sulfone anion coupling of the sulfone 3 with a northern hemisphere aldehyde 2 and subsequent functional group elaboration.

引用

页码：7479 / 7482

页数：4

共 28 条

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