BINDING OF AN IMIDAZOLIDINE (CLONIDINE), AN OXAZOLOAZEPIN (B-HT 933) AND A THIAZOLOAZEPIN (B-HT 920) TO RAT-BRAIN ALPHA-ADRENOCEPTORS AND RELATION TO CARDIOVASCULAR EFFECTS

被引:71
作者
HAMMER, R
KOBINGER, W
PICHLER, L
机构
[1] ERNST BOEHRINGER INST ARZNEIMITTELFORSCH,DEPT PHARMACOL,DR BOEHRINGER GASSE 5-11,A-1121 VIENNA,AUSTRIA
[2] DR KARL THOMAE GMBH,DEPT BIOCHEM,D-7950 BIBERACH,FED REP GER
关键词
D O I
10.1016/0014-2999(80)90095-3
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:277 / 285
页数:9
相关论文
共 16 条
[1]   ALPHA-NORADRENERGIC RECEPTOR-BINDING IN MAMMALIAN BRAIN - DIFFERENTIAL LABELING OF AGONIST AND ANTAGONIST STATES [J].
GREENBERG, DA ;
UPRICHARD, DC ;
SNYDER, SH .
LIFE SCIENCES, 1976, 19 (01) :69-76
[2]   BINDING CHARACTERISTICS OF PRAZOSIN-H-3 TO RAT-BRAIN ALPHA-ADRENERGIC RECEPTORS [J].
GREENGRASS, P ;
BREMNER, R .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 55 (03) :323-326
[3]  
HEINZEL G, 1979, DATA ANAL EVALUATION
[4]  
HOEFKE W, 1975, ARZNEIMITTEL-FORSCH, V25, P786
[6]   PHARMACOLOGICAL CHARACTERIZATION OF B-HT-933 (2-AMINO-6-ETHYL-4,5,7,8-TETRAHYDRO-6H-OXAZOLO-[5,4-D]AZEPIN-DIHYDROCHLORIDE) AS A HYPOTENSIVE AGENT OF CLONIDINE-TYPE [J].
KOBINGER, W ;
PICHLER, L .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1977, 300 (01) :39-46
[7]   INVESTIGATION INTO SOME IMIDAZOLINE COMPOUNDS, WITH RESPECT TO PERIPHERAL ALPHA-ADRENOCEPTOR STIMULATION AND DEPRESSION OF CARDIOVASCULAR CENTERS [J].
KOBINGER, W ;
PICHLER, L .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1975, 291 (02) :175-191
[8]   DIRECT BIOCHEMICAL DEMONSTRATION OF 2 TYPES OF ALPHA-ADRENORECEPTOR IN RAT-BRAIN [J].
MIACH, PJ ;
DAUSSE, JP ;
MEYER, P .
NATURE, 1978, 274 (5670) :492-494
[9]   GENERAL STRATEGY FOR PARAMETER ESTIMATION FROM ISOSTERIC AND ALLOSTERIC-KINETIC DATA AND BINDING MEASUREMENTS [J].
REICH, JG ;
WANGERMANN, G ;
ROHDE, K ;
FALCK, M .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1972, 26 (03) :368-+
[10]  
SCHMITT H, 1977, HDB EXPT PHARMAKOLOG, V39, P299