A SAFE, SIMPLE, ONE-POT PREPARATION OF N-DERIVATIZED BETA-AMINO ALCOHOLS AND OXAZOLIDINONES FROM AMINO-ACIDS

被引：43

作者：

CORREA, A ^{[1
]}

DENIS, JN ^{[1
]}

GREENE, AE ^{[1
]}

机构：

[1] UNIV JOSEPH FOURIER GRENOBLE,LEDSS,BAT 52,F-38041 GRENOBLE,FRANCE

来源：

SYNTHETIC COMMUNICATIONS | 1991年 / 21卷 / 01期

关键词：

D O I：

10.1080/00397919108020783

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

N-tert-Butoxycarbonyl, N-benzoyl, N-benzyloxycarbonyl, and oxazolidinone derivatives of beta-amino alcohols have been prepared from amino acids in 72 to 91 % yields through lithium aluminum hydride reduction followed by in situ derivatization.

引用

页码：1 / 9

页数：9

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