A MILD PREPARATION OF AMINO-ACID N-ACYLSULFONAMIDES

被引：0
作者：
PELLETIER, JC
HESSON, DP
机构：
来源：
SYNLETT | 1995年 / 11期
关键词：
ASPARTIC ACID; GLUTAMIC ACID; ACYLSULFONAMIDES;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A mild preparation of acylsulfonamide amino acids has been devised which is an improvement over existing methods. In particular, gamma-substituted glutamic acid acylsulfonamide derivatives have been prepared without the competitive formation of pyroglutamates.
引用
收藏
页码：1141 / &
相关论文
共 13 条
  • [1] AMINO-ACID SYNTHESIS USING (L)-PYROGLUTAMIC ACID AS A CHIRAL STARTING MATERIAL
    BALDWIN, JE
    MIRANDA, T
    MOLONEY, M
    HOKELEK, T
    [J]. TETRAHEDRON, 1989, 45 (23) : 7459 - 7468
  • [2] NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE .6. DESIGN OF A POTENT, INTRATRACHEALLY ACTIVE, PYRIDONE-BASED TRIFLUOROMETHYL KETONE
    BERNSTEIN, PR
    GOMES, BC
    KOSMIDER, BJ
    VACEK, EP
    WILLIAMS, JC
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (01) : 212 - 215
  • [3] BOLIN DR, 1987, ORG PREP P INT, V21, P67
  • [4] NONPEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGONISTS .2. DESIGN, SYNTHESIS, AND BIOLOGICAL-ACTIVITY OF N-SUBSTITUTED (PHENYLAMINO)PHENYLACETIC ACIDS AND ACYL SULFONAMIDES
    DHANOA, DS
    BAGLEY, SW
    CHANG, RSL
    LOTTI, VJ
    CHEN, TB
    KIVLIGHN, SD
    ZINGARO, GJ
    SIEGL, PKS
    PATCHETT, AA
    GREENLEE, WJ
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1993, 36 (26) : 4239 - 4249
  • [5] DRUMMOND JT, 1988, TETRAHEDRON LETT, V27, P1653
  • [6] HOHENLOHEOEHRIN.K, 1968, MONTASH CHEM, V99, P1301
  • [7] HOHENLOHEOEHRIN.K, 1968, MONTASH CHEM, V99, P1289
  • [8] SYNTHESIS AND STRUCTURE-ACTIVITY STUDIES ON ACIDIC AMINO-ACIDS AND RELATED DIACIDS AS NMDA RECEPTOR LIGANDS
    JOHANSEN, TN
    FRYDENVANG, K
    EBERT, B
    KROGSGAARDLARSEN, P
    MADSEN, U
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (20) : 3252 - 3262
  • [9] LIPTON SA, 1994, NEW ENGL J MED, V330, P613
  • [10] POSSIBLE THERAPEUTIC APPLICATIONS OF ANTAGONISTS OF EXCITATORY AMINO-ACID NEUROTRANSMITTERS
    MELDRUM, B
    [J]. CLINICAL SCIENCE, 1985, 68 (02) : 113 - 122
12