KETANSERIN, A SEROTONERGIC AND ALPHA1-ADRENERGIC ANTAGONIST, BLOCKS CARDIAC NA+ CHANNELS AND LENGTHENS REPOLARIZATION

被引:0
|
作者
KAMIYA, K [1 ]
VENKATESH, N [1 ]
SINGH, BN [1 ]
机构
[1] VET ADM WADSWORTH MED CTR,LOS ANGELES,CA 90073
关键词
D O I
暂无
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:A156 / A156
页数:1
相关论文
共 50 条
  • [21] GATING OF CARDIAC NA+ CHANNELS IN EXCISED MEMBRANE PATCHES AFTER MODIFICATION BY ALPHA-CHYMOTRYPSIN
    VALENZUELA, C
    BENNETT, PB
    BIOPHYSICAL JOURNAL, 1994, 67 (01) : 161 - 171
  • [22] DIFFERENCES IN VASODILATING ACTION BETWEEN KETANSERIN, A 5-HT2-SEROTONERGIC RECEPTOR ANTAGONIST, AND TERAZOSIN, AN ALPHA-1-ADRENOCEPTOR ANTAGONIST, IN ANESTHETIZED RABBITS
    IKEDA, K
    TAKATA, M
    TOMODA, F
    MIKAWA, M
    IIDA, H
    SASAYAMA, S
    JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1987, 10 : S69 - S72
  • [23] Betaxolol, a β1-adrenoceptor antagonist, reduces Na+ influx into cortical synaptosomes by direct interaction with Na+ channels:: comparison with other β-adrenoceptor antagonists
    Chidlow, G
    Melena, J
    Osborne, NN
    BRITISH JOURNAL OF PHARMACOLOGY, 2000, 130 (04) : 759 - 766
  • [24] Enhanced renoprotective effect of angiotensin converting enzyme inhibitor combined with alpha1-adrenergic antagonist in spontaneously hypertensive rats with renal ablation
    Kanazawa, M
    Kohzuki, M
    Kurosawa, H
    Minami, N
    Ito, O
    Saito, T
    Yasujima, M
    Abe, K
    JOURNAL OF HYPERTENSION, 2004, 22 : S38 - S38
  • [25] ALPHA-1 ADRENERGIC ACTIVATION OF THE NA+ PUMP IN VASCULAR SMOOTH-MUSCLE CELLS
    ALLEN, JC
    NAVRAN, SS
    SEIDEL, CL
    FASEB JOURNAL, 1988, 2 (04): : A933 - A933
  • [26] ALPHA-1-ADRENERGIC STIMULATION OF NA-H EXCHANGE IN CARDIAC MYOCYTES
    WALLERT, MA
    FROHLICH, O
    AMERICAN JOURNAL OF PHYSIOLOGY, 1992, 263 (05): : C1096 - C1102
  • [28] BETA-ADRENERGIC MODULATION OF CURRENTS PRODUCED BY RAT CARDIAC NA+ CHANNELS EXPRESSED IN XENOPUS-LAEVIS OOCYTES
    SCHREIBMAYER, W
    FROHNWIESER, B
    DASCAL, N
    PLATZER, D
    SPREITZER, B
    ZECHNER, R
    KALLEN, RG
    LESTER, HA
    RECEPTORS & CHANNELS, 1994, 2 (04): : 339 - 350
  • [29] MOLECULAR CHARACTERIZATION OF CARDIAC NA+ CHANNELS - EXPRESSION OF BRAIN-1 AND A NEW MEMBER OF THE FAMILY OF NA+ CHANNEL GENES IN RAT MYOCARDIUM
    SILLS, MN
    XU, YC
    COOPERMAN, S
    MANDEL, G
    CHIEN, KR
    CLINICAL RESEARCH, 1988, 36 (03): : A318 - A318
  • [30] Alpha1-Adrenergic Receptor Activation Stimulates Calcium Entry and Proliferation via TRPC6 Channels in Cultured Human Mesangial Cells
    Kong, Fanwu
    Ma, Linlin
    Zou, Li
    Meng, Kexin
    Ji, Tianrong
    Zhang, Lei
    Zhang, Rui
    Jiao, Jundong
    CELLULAR PHYSIOLOGY AND BIOCHEMISTRY, 2015, 36 (05) : 1928 - 1938