NEW SYNTHESIS OF 1-SUBSTITUTED 3-(2-AMINOETHYL) INDOLES

被引：2

作者：

GUNGOR, T

MALABRE, P

TEULON, JM

机构：

来源：

SYNTHETIC COMMUNICATIONS | 1994年 / 24卷 / 16期

关键词：

D O I：

10.1080/00397919408019049

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A number of 1 -substituted 3-(2-aminoethyl) indoles were prepared, in one step, by alkylation of the corresponding 3-(2-aminoethyl)indoles (tryptamines) in the presence of NaH.

引用

页码：2247 / 2256

页数：10

共 10 条

[1] TRYPTAMINES, CARBOLINES, AND RELATED COMPOUNDS .2. A CONVENIENT SYNTHESIS OF TRYPTAMINES AND BETA-CARBOLINES [J].

ABRAMOVITCH, RA ;

SHAPIRO, D .

JOURNAL OF THE CHEMICAL SOCIETY, 1956, (NOV) :4589-4592

[2]

BRU N, Patent No. 7832576

[3]

GUNGOR T, UNPUB J MED CHEM

[4] ZUR KENNTNIS DER TETRAHYDROCARBOLIN-VERBINDUNGEN .1. [J].

HORLEIN, U .

CHEMISCHE BERICHTE-RECUEIL, 1954, 87 (04) :463-472

[5]

JULIA M, 1965, B SOC CHIM FR, V5, P1411

[6]

KALIR A, 1966, J MED CHEM, P793

[7] A CONVENIENT SYNTHESIS OF TRYPTAMINES [J].

MEROUR, JY ;

BUZAS, A .

SYNTHETIC COMMUNICATIONS, 1988, 18 (18) :2331-2335

[8]

SHAW EN, 1956, J PHARMACOL EXP THER, V116, P164

[9] SYNTHESIS + PHARMACOLOGY OF SOME BETA-SPIROINDOLENINES + INDOLINES [J].

WEISBACH, JA ;

CAVA, MP ;

DOUGLAS, B ;

DESANCTIS, NJ ;

MACKO, E .

JOURNAL OF MEDICINAL CHEMISTRY, 1964, 7 (06) :735-&

[10]

1953, Patent No. 2642438

← 1 →