[H-3] DOMPERIDONE LABELS ONLY A SINGLE POPULATION OF RECEPTORS WHICH CONVERT FROM HIGH TO LOW AFFINITY FOR DOPAMINE IN RAT-BRAIN

被引:24
作者
GRIGORIADIS, D
SEEMAN, P
机构
关键词
D O I
10.1007/BF00633192
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:21 / 25
页数:5
相关论文
共 18 条
[1]   DOMPERIDONE-H-3 - SELECTIVE LIGAND FOR DOPAMINE RECEPTORS [J].
BAUDRY, M ;
MARTRES, MP ;
SCHWARTZ, JC .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 308 (03) :231-237
[2]  
FLEMING WW, 1972, J PHARMACOL-PARIS, V181, P339
[3]   DOPAMINE D2-RECEPTORS IN THE ANTERIOR-PITUITARY - A SINGLE POPULATION WITHOUT RECIPROCAL ANTAGONIST AGONIST STATES [J].
GEORGE, SR ;
WATANABE, M ;
SEEMAN, P .
JOURNAL OF NEUROCHEMISTRY, 1985, 44 (04) :1168-1177
[4]   THE DOPAMINE NEUROLEPTIC RECEPTOR [J].
GRIGORIADIS, D ;
SEEMAN, P .
CANADIAN JOURNAL OF NEUROLOGICAL SCIENCES, 1984, 11 (01) :108-113
[5]  
GRIGORIADIS D, 1985, J NEUROCHEM, V44, P1929
[6]   INTERACTIONS OF AGONISTS WITH D-2 DOPAMINE-RECEPTORS - EVIDENCE FOR A SINGLE RECEPTOR POPULATION EXISTING IN MULTIPLE AGONIST AFFINITY-STATES IN RAT STRIATAL MEMBRANES [J].
HAMBLIN, MW ;
LEFF, SE ;
CREESE, I .
BIOCHEMICAL PHARMACOLOGY, 1984, 33 (06) :877-887
[7]   QUANTITATIVE-DETERMINATION OF DOPAMINE RECEPTOR SUBTYPES NOT LINKED TO ACTIVATION OF ADENYLATE-CYCLASE IN RAT STRIATUM [J].
HUFF, RM ;
MOLINOFF, PB .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1982, 79 (23) :7561-7565
[8]   COMPARISON OF INVITRO AND INVIVO DOPAMINE RECEPTOR ANTAGONISM PRODUCED BY SUBSTITUTED BENZAMIDE DRUGS [J].
JENNER, P ;
ELLIOTT, PNC ;
CLOW, A ;
REAVILL, C ;
MARSDEN, CD .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1978, 30 (01) :46-48
[9]   EFFECTS OF GTP ON H-3-LABELED DOMPERIDONE BINDING AND ITS DISPLACEMENT BY DOPAMINE IN RAT STRIATAL HOMOGENATES [J].
LAZARENO, S .
JOURNAL OF RECEPTOR RESEARCH, 1983, 3 (1-2) :163-175
[10]   SPIPERONE - LIGAND OF CHOICE FOR NEUROLEPTIC RECEPTORS .1. KINETICS AND CHARACTERISTICS OF INVITRO BINDING [J].
LEYSEN, JE ;
GOMMEREN, W ;
LADURON, PM .
BIOCHEMICAL PHARMACOLOGY, 1978, 27 (03) :307-316