AGONISTS, INVERSE AGONISTS, AND ANTAGONISTS OF BENZODIAZEPINE RECEPTORS

被引:1
|
作者
HAEFELY, WE [1 ]
机构
[1] F HOFFMANN LA ROCHE & CO LTD,PHARMACEUT RES,CH-4002 BASEL,SWITZERLAND
关键词
D O I
10.1016/0014-2999(90)91286-K
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:38 / 38
页数:1
相关论文
共 50 条
  • [21] COMFA APPROACH TO LONG-LIVED INVERSE AGONISTS AT BENZODIAZEPINE RECEPTORS
    ALLEN, MS
    HAGEN, TJ
    KOEHLER, K
    COOK, JM
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1990, 200 : 93 - MEDI
  • [23] Agonists, inverse agonists, and antagonists as therapeutic approaches to manipulate retinoic acid-related orphan receptors
    Nematisouldaragh, Darya
    Nguyen, Huong
    Rabinovich-Nikitin, Inna
    CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 2024, 102 (11) : 620 - 633
  • [24] THE EFFECT OF BENZODIAZEPINE AGONISTS AND INVERSE AGONISTS IN A RAT-FEEDING MODEL
    DEACON, RMJ
    MCCULLOCH, AJ
    GARDNER, CR
    PSYCHOPHARMACOLOGY, 1986, 89 (04) : S56 - S56
  • [25] BIDIRECTIONAL EFFECTS OF CHRONIC TREATMENT WITH AGONISTS AND INVERSE AGONISTS AT THE BENZODIAZEPINE RECEPTOR
    LITTLE, HJ
    NUTT, DJ
    TAYLOR, SC
    BRAIN RESEARCH BULLETIN, 1987, 19 (03) : 371 - 378
  • [26] Chronic agonist treatment converts antagonists into inverse agonists at δ-opioid receptors
    Liu, JG
    Prather, PL
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2002, 302 (03): : 1070 - 1079
  • [27] BIOMIMETIC APPROACH TO POTENTIAL BENZODIAZEPINE AGONISTS AND ANTAGONISTS
    CAIN, M
    GUZMAN, F
    COOK, JM
    RICE, KC
    SKOLNICK, P
    HETEROCYCLES, 1982, 19 (06) : 1003 - 1007
  • [28] Psychotogenic properties of benzodiazepine receptor inverse agonists
    Sarter, M
    Bruno, JP
    Berntson, GG
    PSYCHOPHARMACOLOGY, 2001, 156 (01) : 1 - 13
  • [29] Psychotogenic properties of benzodiazepine receptor inverse agonists
    Martin Sarter
    John P. Bruno
    Gary G. Berntson
    Psychopharmacology, 2001, 156 : 1 - 13
  • [30] DISTINCTION OF BENZODIAZEPINE RECEPTOR AGONISTS AND INVERSE AGONISTS BY BINDING-STUDIES INVITRO
    KAROBATH, M
    SUPAVILAI, P
    BOREA, PA
    ADVANCES IN BIOCHEMICAL PSYCHOPHARMACOLOGY, 1983, 38 : 37 - 45