AGONISTS, INVERSE AGONISTS, AND ANTAGONISTS OF BENZODIAZEPINE RECEPTORS

被引:1
|
作者
HAEFELY, WE [1 ]
机构
[1] F HOFFMANN LA ROCHE & CO LTD,PHARMACEUT RES,CH-4002 BASEL,SWITZERLAND
关键词
D O I
10.1016/0014-2999(90)91286-K
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:38 / 38
页数:1
相关论文
共 50 条
  • [1] THIENYLPYRAZOLOQUINOLINES - POTENT AGONISTS AND INVERSE AGONISTS TO BENZODIAZEPINE RECEPTORS
    TAKADA, S
    SHINDO, H
    SASATANI, T
    CHOMEI, N
    MATSUSHITA, A
    EIGYO, M
    KAWASAKI, K
    MURATA, S
    TAKAHARA, Y
    SHINTAKU, H
    JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (09) : 1738 - 1745
  • [2] INVITRO CHARACTERIZATION OF BENZODIAZEPINE RECEPTOR AGONISTS, ANTAGONISTS, INVERSE AGONISTS AND AGONIST ANTAGONISTS
    WOOD, PL
    LOO, P
    BRAUNWALDER, A
    YOKOYAMA, N
    CHENEY, DL
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1984, 231 (03): : 572 - 576
  • [3] INTERACTION OF BENZODIAZEPINE AGONISTS AND ANTAGONISTS WITH DIFFERENT BENZODIAZEPINE RECEPTORS
    SIEGHART, W
    DREXLER, G
    MAYER, A
    SCHUSTER, A
    ADVANCES IN BIOCHEMICAL PSYCHOPHARMACOLOGY, 1983, 38 : 11 - 19
  • [4] BENZODIAZEPINE RECEPTORS - MODE OF INTERACTION OF AGONISTS AND ANTAGONISTS
    MOHLER, H
    ADVANCES IN BIOCHEMICAL PSYCHOPHARMACOLOGY, 1983, 37 : 247 - 254
  • [5] INVERSE AGONISTS AND ANTAGONISTS OF RETINOID RECEPTORS
    Bourguet, William
    de Lera, Angel R.
    Gronemeyer, Hinrich
    METHODS IN ENZYMOLOGY, VOLUME 485: CONSTITUTIVE ACTIVITY IN RECEPTORS AND OTHER PROTEINS, PART B, 2010, 485 : 161 - 195
  • [7] ACTIONS AND INTERACTIONS OF BENZODIAZEPINE AGONISTS, ANTAGONISTS AND INVERSE AGONISTS ON SUPRAHYOID MUSCLE TWITCHING
    JAMES, V
    GARDNER, CR
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 113 (02) : 233 - 238
  • [8] CONFORMATIONAL SHIFTS AT THE BENZODIAZEPINE RECEPTOR RELATED TO THE BINDING OF AGONISTS ANTAGONISTS AND INVERSE AGONISTS
    FRYER, RI
    COOK, C
    GILMAN, NW
    WALSER, A
    LIFE SCIENCES, 1986, 39 (21) : 1947 - 1957
  • [9] EFFECTS OF BENZODIAZEPINE AGONISTS, ANTAGONISTS AND INVERSE AGONISTS ON MOUSE PUP ULTRASONIC CALLING
    NASTITI, K
    BENTON, D
    BRAIN, PF
    AGGRESSIVE BEHAVIOR, 1989, 15 (01) : 92 - 92
  • [10] PHARMACODYNAMIC INTERACTIONS BETWEEN MIDAZOLAM AND BENZODIAZEPINE PARTIAL AGONISTS, ANTAGONISTS AND INVERSE AGONISTS
    MANDEMA, JW
    KUCK, MT
    DANHOF, M
    CLINICAL PHARMACOLOGY & THERAPEUTICS, 1991, 49 (02) : 125 - 125