TUMOR-PROMOTING AND HYPERPLASTIC EFFECTS OF PHORBOL AND DAPHNANE ESTERS IN CD-1 MOUSE SKIN AND A SYNERGISTIC EFFECT OF CALCIUM IONOPHORE WITH THE NON-PROMOTING ACTIVATOR OF PROTEIN KINASE-C, SAPINTOXIN-A

被引:33
作者
BROOKS, G
EVANS, AT
AITKEN, A
EVANS, FJ
机构
[1] UNIV LONDON,SCH PHARM,DEPT PHARMACOGNOSY,29-39 BRUNSWICK SQ,LONDON WC1N 1AX,ENGLAND
[2] NATL INST MED RES,PROT STRUCT LAB,LONDON NW7 1AA,ENGLAND
关键词
D O I
10.1093/carcin/10.2.283
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:283 / 288
页数:6
相关论文
共 28 条
[1]  
ALBERT PR, 1985, J BIOL CHEM, V260, P87146
[2]  
BERKELHAMMER J, 1987, CANCER RES, V47, P1251
[3]   TOXIC PHORBOL ESTERS FROM CHINESE TALLOW STIMULATE PROTEIN-KINASE-C [J].
BROOKS, G ;
MORRICE, NA ;
ELLIS, C ;
AITKEN, A ;
EVANS, AT ;
EVANS, FJ .
TOXICON, 1987, 25 (11) :1229-1233
[4]  
BROOKS G, 1987, Journal of Pharmacy and Pharmacology, V39, p98P
[5]   SAPINTOXIN-A - A FLUORESCENT PHORBOL ESTER THAT IS A POTENT ACTIVATOR OF PROTEIN KINASE-C BUT IS NOT A TUMOR PROMOTER [J].
BROOKS, G ;
EVANS, AT ;
AITKEN, A ;
EVANS, FJ .
CANCER LETTERS, 1987, 38 (1-2) :165-170
[6]   THE STIMULATION OF PHOSPHORYLATION OF INTRACELLULAR PROTEINS IN GH3-RAT PITUITARY-TUMOR CELLS BY PHORBOL ESTERS OF DISTINCT BIOLOGICAL-ACTIVITY [J].
BROOKS, SF ;
EVANS, FJ ;
AITKEN, A .
FEBS LETTERS, 1987, 224 (01) :109-116
[7]  
BROOKS SF, 1988, IN PRESS EUR J BIOCH
[8]   FURTHER OBSERVATIONS ON THE EFFECT OF CALCIUM IONOPHORES ON ASCITES TUMOR-CELLS [J].
CALVIELLO, G ;
BOSSI, D ;
CITTADINI, A .
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 1987, 259 (01) :38-45
[9]  
EDWARDS MC, 1983, ACTA PHARMACOL TOX, V53, P177
[10]  
Ellis C. A., 1987, PHYTOTHER RES, V1, P187