(Z)-2-(2,4-DICHLOROPHENOXY)METHYL-3-FLUOROALLYLAMINE (MDL 72638) - A CLORGYLINE ANALOG WITH SURPRISING SELECTIVITY FOR MONOAMINE-OXIDASE TYPE-B

被引：10

作者：

MCDONALD, IA ^{[1
]}

PALFREYMAN, MG ^{[1
]}

ZREIKA, M ^{[1
]}

BEY, P ^{[1
]}

机构：

[1] MERRELL DOW RES INST,STRASBOURG CTR,F-67084 STRASBOURG,FRANCE

来源：

BIOCHEMICAL PHARMACOLOGY | 1986年 / 35卷 / 02期

关键词：

D O I：

10.1016/0006-2952(86)90538-1

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：349 / 351

页数：3

共 14 条

[1] (E)-2-(3,4-DIMETHOXYPHENYL)-3-FLUOROALLYLAMINE - A SELECTIVE, ENZYME-ACTIVATED INHIBITOR OF TYPE-B MONOAMINE-OXIDASE
BEY, P
FOZARD, J
LACOSTE, JM
MCDONALD, IA
ZREIKA, M
PALFREYMAN, MG
JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (01) : 9 - 10
[2] INHIBITION OF MONOAMINE-OXIDASE BY THE R-ENANTIOMER AND S-ENANTIOMER OF N[3-(2,4-DICHLOROPHENOXY)PROPYL]-N-METHYL-3-BUTYN-2-AMINE
DOSTERT, P
OBRIEN, EM
TIPTON, KF
MERONI, M
MELLONI, P
BENEDETTI, MS
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 1992, 27 (01) : 45 - 52
[3] INHIBITION OF TYPE-A AND TYPE-B MONOAMINE-OXIDASE BY 1-METHYL-4-PHENYL-1,2,3,6-TETRAHYDROPYRIDINE
FULLER, RW
HEMRICKLUECKE, SK
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1985, 232 (03): : 696 - 701
[4] INHIBITION OF A TYPE-B MONOAMINE-OXIDASE INHIBITOR, (E)-2-(4-FLUOROPHENETHYL)-3-FLUOROALLYLAMINE (MDL-72974A), ON SEMICARBAZIDE-SENSITIVE AMINE OXIDASES ISOLATED FROM VASCULAR TISSUES AND SERA OF DIFFERENT SPECIES
YU, PH
ZUO, DM
BIOCHEMICAL PHARMACOLOGY, 1992, 43 (02) : 307 - 312
[5] A REACTIVE METABOLITE OF 1-METHYL-4-PHENYL-1,2,3,6-TETRAHYDROPYRIDINE IS FORMED IN RAT-BRAIN INVITRO BY TYPE-B MONOAMINE-OXIDASE
CORSINI, GU
PINTUS, S
BOCCHETTA, A
PICCARDI, MP
DELZOMPO, M
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1986, 238 (02): : 648 - 652
[6] INHIBITION OF TYPE-A AND TYPE-B MONOAMINE-OXIDASE BY 6,7-DIHYDROXY-1,2,3,4-TETRAHYDROISOQUINOLINES AND THEIR N-METHYLATED DERIVATIVES
MINAMI, M
MARUYAMA, W
DOSTERT, P
NAGATSU, T
NAOI, M
JOURNAL OF NEURAL TRANSMISSION-GENERAL SECTION, 1993, 92 (2-3) : 125 - 135
[7] PHOTOINACTIVATION OF B-TYPE MONOAMINE-OXIDASE BY A 1-METHYL-4-PHENYL-1,2,3,6-TETRAHYDROPYRIDINE METABOLITE
BUCKMAN, TD
EIDUSON, S
JOURNAL OF BIOLOGICAL CHEMISTRY, 1985, 260 (22) : 1899 - 1902
[8] INHIBITION OF MONOAMINE-OXIDASE TYPE-A AND TYPE-B BY 2-ARYL-4H-1,3,4-OXADIAZIN-5(6H)-ONE DERIVATIVES
MAZOUZ, F
LEBRETON, L
MILCENT, R
BURSTEIN, C
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 1988, 23 (05) : 441 - 451
[9] CONVERSION OF THE NEUROTOXIC PRECURSOR 1-METHYL-4-PHENYL-1,2,5,6-TETRAHYDROPYRIDINE INTO ITS PYRIDINIUM METABOLITE BY HUMAN-PLATELET MONOAMINE-OXIDASE TYPE-B
DAPRADA, M
CESURA, AM
KETTLER, R
ZURCHER, G
HAEFELY, WE
NEUROSCIENCE LETTERS, 1985, 57 (03) : 257 - 262
[10] 5-ARYL-1,3,4-OXADIAZOL-2(3H)-ONE DERIVATIVES AND SULFUR ANALOGS AS NEW SELECTIVE AND COMPETITIVE MONOAMINE-OXIDASE TYPE-B INHIBITORS
MAZOUZ, F
LEBRETON, L
MILCENT, R
BURSTEIN, C
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 1990, 25 (08) : 659 - 671

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