IRREVERSIBLE OPIATE AGONISTS AND ANTAGONISTS .5. HYDRAZONE AND ACYLHYDRAZONE DERIVATIVES OF NALTREXONE

被引:48
作者
LUKE, MC
HAHN, EF
PRICE, M
PASTERNAK, GW
机构
[1] CORNELL UNIV,MED CTR,COLL MED,DEPT NEUROL,NEW YORK,NY 10021
[2] CORNELL UNIV,MED CTR,COLL MED,DEPT PHARMACOL,NEW YORK,NY 10021
[3] ROCKEFELLER UNIV,BIOCHEM ENDOCRINOL LAB,NEW YORK,NY 10021
关键词
D O I
10.1016/0024-3205(88)90215-9
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:1249 / 1256
页数:8
相关论文
共 9 条
[1]  
CLARK JA, IN PRESS MOL PHARM
[2]  
HAHN EF, 1985, J PHARMACOL EXP THER, V235, P846
[3]   NALOXONAZINE, A POTENT, LONG-LASTING INHIBITOR OF OPIATE BINDING-SITES [J].
HAHN, EF ;
PASTERNAK, GW .
LIFE SCIENCES, 1982, 31 (12-1) :1385-1388
[4]  
HAHN EF, 1982, J NEUROSCI, V2, P572
[5]  
HAHN EF, 1985, J PHARMACOL EXP THER, V235, P839
[6]   NALOXONAZINE ACTIONS INVIVO [J].
LING, GSF ;
SIMANTOV, R ;
CLARK, JA ;
PASTERNAK, GW .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 129 (1-2) :33-38
[7]   MINIREVIEW - MULTIPLE MU OPIATE RECEPTORS [J].
PASTERNAK, GW ;
WOOD, PJ .
LIFE SCIENCES, 1986, 38 (21) :1889-1898
[8]  
PASTERNAK GW, 1980, J MED CHEM, V23, P674, DOI 10.1021/jm00180a019
[9]  
PRICE M, IN PRESS MOL PHARM