DIPEPTIDE ANALOGS - SYNTHESIS OF A POTENT RENIN INHIBITOR

被引：31

作者：

BOCK, MG

DIPARDO, RM

EVANS, BE

RITTLE, KE

BOGER, JS

FREIDINGER, RM

VEBER, DF

机构：

来源：

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1985年 / 03期

关键词：

D O I：

10.1039/c39850000109

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

引用

页码：109 / 110

页数：2

共 8 条

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STABILITO, II ;

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RICH, DH ;

BOPARI, AS .

NATURE, 1983, 303 (5912) :81-84

[2]

BOGER J, 1983, PEPTIDES STRUCTURE F, P569

[3] (2S,3S,4R)-4-AMINO-3-HYDROXY-2-METHYLPENTANOIC ACID - ENANTIOSELECTIVE SYNTHESIS OF AN AMINO-ACID CONSTITUENT OF BLEOMYCIN [J].

DIPARDO, RM ;

BOCK, MG .

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[4] ENANTIOSELECTIVE ALDOL CONDENSATIONS .2. ERYTHRO-SELECTIVE CHIRAL ALOL CONDENSATIONS VIA BORON ENOLATES [J].

EVANS, DA ;

BARTROLI, J ;

SHIH, TL .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1981, 103 (08) :2127-2129

[5] SYNTHESIS OF HYDROXYETHYLENE AND KETOMETHYLENE DIPEPTIDE ISOSTERES [J].

HOLLADAY, MW ;

RICH, DH .

TETRAHEDRON LETTERS, 1983, 24 (41) :4401-4404

[6] KINETICS OF REACTION OF RENIN WITH 9 SYNTHETIC PEPTIDE SUBSTRATES [J].

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HOCHSTRASSER, H .

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[7]

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[8]

VEBER DF, 1984, T BIOCH SOC

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